| Company Name: |
3B Pharmachem (Wuhan) International Co.,Ltd.
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| Tel: |
821-50328103-801 18930552037 |
| Email: |
3bsc@sina.com |
| Products Intro: |
Product Name:Proxyfan oxalate;4-[3-(PhenylMethoxy)propyl]-1H-iMidazoleoxalate
CAS:177708-09-7
Purity:99% HPLC Package:1Mg ; 5Mg;10Mg ;100Mg;250Mg ;500Mg ;1g;2.5g ;5g ;10g
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| Company Name: |
BOC Sciences
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| Tel: |
1-631-485-4226; 16314854226 |
| Email: |
info@bocsci.com |
| Products Intro: |
Product Name:Proxyfan maleate
CAS:177708-09-7
Purity:98% by HPLC Remarks:Proxyfan oxalate is a high affinity histamine H3 receptor ligand (pKi = 8.62), acting as a protean agonist with activity ranges from full agonist to inverse agonist depending on system used.
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| | PROXYFAN MALEATE Basic information |
| Product Name: | PROXYFAN MALEATE | | Synonyms: | PROXYFAN MALEATE;4-[3-(Phenylmethoxy)propyl]-1H-imidazoleoxalate;Proxyfan oxalate;1H-Imidazole, 5-[3-(phenylmethoxy)propyl]- | | CAS: | 177708-09-7 | | MF: | C13H16N2O | | MW: | 216.28 | | EINECS: | | | Product Categories: | | | Mol File: | 177708-09-7.mol |  |
| | PROXYFAN MALEATE Chemical Properties |
| Boiling point | 414.5±33.0 °C(Predicted) | | density | 1.115±0.06 g/cm3(Predicted) | | storage temp. | Desiccate at RT | | solubility | Soluble to 100 mM in DMSO and to 100 mM in water | | form | Powder | | pka | 14.60±0.10(Predicted) |
| | PROXYFAN MALEATE Usage And Synthesis |
| Biological Activity | High affinity histamine H 3 receptor ligand (pK i = 8.62) that acts as a protean agonist at recombinant and native receptors. In functional studies, activity ranges from full agonist to inverse agonist depending on system used. Displays partial agonist effects on cAMP inhibition and MAPK activity, neutral antagonist activity on histamine release and partial inverse agonism of [ 3 H]-arachidonic acid release. |
| | PROXYFAN MALEATE Preparation Products And Raw materials |
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