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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
2-[6-(2,5-dichloropyrimidin-4-yl)-4-fluoro-1-isopropyl-benzimidazol-2-yl]propan-2-ol 2380323-09-9 详细
3-phenoxycyclobutanecarboxylic acid 3-苯氧基 - 环丁烷羧酸 1263284-46-3 详细
tert-butyl 4-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]piperidine-1-carboxylate 4-(1-BOC-4-哌啶基)苯硼酸频哪醇酯 956136-85-9 详细
5-[(3,5-difluorophenyl)methyl]-1H-indazol-3-amine 5-(3,5-二氟苄基)-1H-吲唑-3-胺 1108745-30-7 详细
cis-1-methyl-3-phenyl-cyclobutanamine;hydrochloride 2702358-29-8 详细
4-[(6-chloro-2-pyridyl)oxymethyl]-3-fluoro-benzonitrile 4-(((6-氯吡啶-2-基)氧基)甲基)-3-氟苄腈 2230200-58-3 详细
4-{3,9-diazaspiro[5.5]undecan-3-yl}-2-methoxyaniline 4-{3,9-二氮杂螺[5.5]十一烷-3-基}-2-甲氧基苯胺 2007917-26-0 详细
2-bromo-6-(6-cyclopropyl-8-fluoro-1-oxo-2-isoquinolyl)benzaldehyde 2-溴-6-[6-环丙基-8-氟-1-氧代异喹啉-2(1H)-基]苯甲醛 1642290-28-5 详细
2-cyclobutylmorpholine 2-环丁基吗啉 1219844-05-9 详细
tert-butyl N-[1-(5-bromo-2-pyridyl)-4-piperidyl]carbamate 叔-丁基 N-[1-(5-溴-2-吡啶基)-4-哌啶基]氨基甲酯 1042917-47-4 详细
3-chloro-4-cyclopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenol 3-氯-4-环丙基-5-(4,4,5,5-四甲基-1,3,2-二氧杂硼-2-基)苯酚 2773311-45-6 详细
(3R)-3-benzyl-1-[(tert-butoxy)carbonyl]piperidine-3-carboxylic acid 阿拉莫林中间体 339539-81-0 详细
2-(3-chloro-4-fluorophenyl)-4,4-dimethyl-1,2,3,4-tetrahydroquinoline-6-carboxylic acid 2-(3-氯-4-氟苯基)-4,4-二甲基-1,2,3,4-四氢喹啉-6-羧酸 1353971-43-3 详细
5-bromo-6-methyl-1-{[2-(trifluoromethyl)phenyl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione 5-溴-6-甲基-1-{[2-(三氟甲基)苯基]甲基}-1,2,3,4-四氢嘧啶-2,4-二酮 2102411-35-6 详细
tert-butyl 3-{[(4-bromophenyl)methyl]amino}azetidine-1-carboxylate 叔-丁基 3-{[(4-溴苯基)甲基]氨基}吖丁啶-1-甲酸基酯 887579-73-9 详细
6-chloro-1-[(1R)-1-(2,4-dichlorophenyl)ethyl]-3-methyl-pyrazolo[3,4-b]pyrazine 2174940-57-7 详细
3-Pyrrolidinecarbonitrile, 1-[3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]- 2304631-52-3 详细
4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)aniline 4-[(4-甲基哌嗪-1-基)甲基]-3-(三氟甲基)苯胺 694499-26-8 详细
3-[[(3S)-4-(difluoromethyl)-2,2-difluoro-3-hydroxy-1,1-dioxo-3H-benzothiophen-5-yl]oxy]-5-fluoro-benzonitrile 1799948-37-0 详细
3-(2,4-dioxohexahydropyrimidin-1-yl)benzoic acid 3-(2,4-二氧四氢嘧啶-1(2H)基)苯甲酸 2377644-59-0 详细
1-cyclopropylcyclopropanecarboxylic acid 1,1'-联(环丙烷)]-1-羧酸 60629-92-7 详细
4-cyclohexyl-3-(trifluoromethyl)phenyl]methanol 4-环己基-3-(三氟甲基)苯基]甲醇 957205-23-1 详细
tert-butyl 4-(6-cyano-2-pyridyl)piperazine-1-carboxylate 4-(6-氰基吡啶-2-基)哌嗪-1-羧酸甲酯 叔丁酯 1461715-72-9 详细
1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxylic acid 4-安替比林羧酸 83-10-3 详细
methyl 4-fluoro-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoate 甲基 4-氟-2-{1H-吡咯并[2,3-b]吡啶-5-氧基}苯酸盐 1235865-75-4 详细
1-(azetidin-3-yl)imidazole dihydrochloride 1-(氮杂环丁烷-3-基)-1H-咪唑盐酸盐 153836-44-3 详细
3-(1-tert-butoxycarbonylazetidin-3-yl)cyclobutanecarboxylic acid 3-(1-(叔丁氧基羰基)氮杂环丁烷-3-基)环丁烷羧酸 1989659-47-3 详细
2-bromo-N-{3-[(4-methoxyphenyl)methoxy]phenyl}thieno[3,2-b]pyridin-7-amine 2-溴-N-{3-[(4-甲氧苯基)甲氧基]苯基}噻吩并[3,2-b]吡啶-7-胺 1228102-89-3 详细
4-(4-chloroquinazolin-7-yl)morpholine 4-(4-氯喹唑啉-7-基)吗啉 1334602-74-2 详细
1-methyl-4-(oxetan-3-yl)piperazine 1-甲基-4-(噁丁环烷-3-基)哌嗪 1788043-99-1 详细
tert-butyl cis-3-(2,6-dichloropyridine-4-carbonyl)cyclobutanecarboxylate 2703696-90-4 详细
4-methyl-4-phenyl-piperidine;hydrochloride 4-甲基-4-苯基哌啶盐酸盐 83949-37-5 详细
1-phenylpiperidin-4-one 1-苯基-4-哌啶酮 19125-34-9 详细
4-(chloromethyl)-5-cyclopropyl-3-(2,6-dichlorophenyl)-1,2-oxazole 4-(氯甲基)-5-环丙基-3-(2,6-二氯苯基)-1,2-噁唑 1268245-50-6 详细
ethyl 1-(1H-pyrazol-3-yl)cyclopropanecarboxylate 2386967-78-6 详细
(4-cyclopropoxyphenyl)boronic acid 4-环丙氧基苯硼酸 871829-90-2 详细
2-[(1R)-1-aminoethyl]-N-[5-chloro-4-(trifluoromethyl)pyridin-2-yl]-1,3-thiazole-5-carboxamide (R)-2-(1-氨基乙基)-N-(5-氯-4-(三氟甲基)吡啶-2-基)噻唑-5-甲酰胺 1095823-62-3 详细
4-(morpholin-4-yl)aniline 4-(吗啉-4-基)苯胺 2524-67-6 详细
(1-cyclopropylcyclopropyl)methanol {[1,1'-联(环丙烷)]-1-基}甲醇 177719-30-1 详细
(3R)-3-methyl-4-(6-nitro-3-pyridyl)morpholine (3R)-3-methyl-4-(6-nitro-3-pyridyl)morpholine 2375165-76-5 详细
(1R,2R)-2-(3-fluoro-4-methoxy-phenyl)cyclopropanecarboxylic acid 220352-90-9 详细
tert-butyl 4-(4-iodo-1H-pyrazol-1-yl)piperidine-1-carboxylate 4-(4-碘-1H-吡唑-1-基)-1-哌啶羧酸-1,1-二甲基乙酯 877399-73-0 详细
(2R,3R,4S,5R)-2-(6-amino-2-chloro-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol (2R,3R,4S,5R)-2-(6-氨基-2-氯-9H-嘌呤-9-基)-5-(羟甲基)噁戊环-3,4-二醇 146-77-0 详细
1-(oxan-4-yl)-1H-pyrazol-4-amine 1-(噁烷-4-基)-1H-吡唑-4-胺 1190380-49-4 详细
4-amino-1-[(3R)-1-[(tert-butoxy)carbonyl]piperidin-3-yl]-1H-pyrazolo[3,4-d]pyrimidine-3-carboxylic acid 4-amino-1-[(3R)-1-[(tert-butoxy)carbonyl]piperidin-3-yl]-1H-pyrazolo[3,4-d]pyrimidine-3-carboxylic acid 1654728-11-6 详细
ethyl trans-2-(2-pyridyl)cyclopropanecarboxylate 58620-63-6 详细
6-cyclopentyl-2-oxo-1,2-dihydropyridine-4-carboxylic acid 6-环戊基-2-氧亚基-1,2-二氢吡啶-4-羧酸 1368348-22-4 详细
ethyl trans-2-(6-bromo-3-pyridyl)cyclopropanecarboxylate 乙基 (1S,2S)-rel-2-(6-溴吡啶-3-基)环丙烷-1-甲酸基酯 1357247-47-2 详细
trans-2-(4-hydroxyphenyl)cyclopropane-1-carboxylic acid (1S,2S)-rel-2-(4-羟基苯基)环丙烷-1-羧酸 731810-73-4 详细
tert-butyl 4-[3-(hydroxymethyl)phenyl]piperidine-1-carboxylate 909422-39-5 909422-39-5 详细
3-bromo-6-cyclopropyl-pyridin-2-amine 3-溴-6-环丙基-吡啶-2-胺 1508445-19-9 详细
2-{2-methyl-5-[4-(methylsulfanyl)phenyl]-1H-pyrrol-1-yl}ethan-1-ol 2-{2-甲基-5-[4-(甲基巯基)苯基]-1H-吡咯-1-基}乙烷-1-醇 494850-27-0 详细
(1R)-1-[4-chloro-2-(3-methyl-1H-pyrazol-1-yl)phenyl]-2,2,2-trifluoroethan-1-ol (1R)-1-[4-氯-2-(3-甲基-1H-吡唑-1-取代)苯基]-2,2,2-三氟乙基-1-醇 1033805-26-3 详细
1-(6-bromo-7-fluoro-1-methyl-indazol-3-yl)hexahydropyrimidine-2,4-dione 1-(6-溴-7-氟-1-甲基-1H-吲唑-3-基)-1,3-二嗪烷-2,4-二酮 2760849-95-2 详细
(2R)-2-phenylpyrrolidine (2R)-2-苯基吡咯烷 56523-47-8 详细
4-[(2,4-diaminopteridin-6-yl)methylamino]benzoic acid;sodium salt 钠 4-{[(2,4-二氨基蝶啶-6-基)甲基]氨基}苯酸盐 100929-45-1 详细
7-[4-(trifluoromethoxy)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-5-one 7-[4-(三氟甲氧基)苯基]-2,3,4,5-四氢-1,4-苯并噁吖庚英-5-酮 1430092-39-9 详细
3-(3-fluoro-2-methoxy-phenyl)isoxazol-5-amine 1465812-19-4 详细
trans-2-(3-ethoxy-4-fluoro-phenyl)cyclopropanamine;hydrochloride (1S,2R)-rel-2-(3-乙氧基-4-氟苯基)环丙烷-1-胺盐酸 2055841-10-4 详细
(2S,3R)-1-(9H-fluoren-9-ylmethoxycarbonyl)-3-phenyl-pyrrolidine-2-carboxylic acid FMOC-(2S,3R)-3-苯基吡咯烷-2-羧酸 281655-32-1 详细
2-[2-(2,6-dioxo-3-piperidyl)-1,3-dioxo-isoindolin-4-yl]oxyacetic acid 2-((2-(2,6-DIOXOPIPERIDIN-3-YL)-1,3-DIOXOISOINDOLIN-4-YL]OXY]ACETIC ACID 1061605-21-7 详细
tert-butyl 4-(5-bromopyridin-2-yl)piperazine-1-carboxylate 4-BOC-1-(5-溴-2-吡啶基)哌嗪 153747-97-8 详细
trans-2-[4-(oxan-2-yloxy)phenyl]cyclopropane-1-carboxylic acid 反-2-[4-(噁烷-2-氧基)苯基]环丙烷-1-羧酸 1946017-75-9 详细
3-cyclohexylazetidine hydrochloride 3-cyclohexylazetidine hydrochloride 7606-38-4 详细
(2E)-1-(1H-1,3-benzodiazol-2-yl)-3-(3-methoxyphenyl)prop-2-en-1-one (E)-1-(2-苯并咪唑基)-3-(3-甲氧基苯基)-2-丙烯-1-酮 1372406-51-3 详细
3-(2,6-difluorophenyl)azetidin-3-ol hydrochloride 2306275-02-3 详细
4-(dimethylamino)-4-(3-fluorophenyl)cyclohexan-1-one 4-(二甲氨基)-4-(3-氟苯基)环己烷-1-酮 863514-54-9 详细
6-bromo-2-chloro-8-cyclopentyl-5-methyl-7H,8H-pyrido[2,3-d]pyrimidin-7-one 6-溴-2-氯-8-环戊基-5-甲基-7H,8H-吡啶并[2,3-d]嘧啶-7-酮 1016636-76-2 详细
3-phenylcyclobutane-1-carboxylic acid 3-苯基环丁烷-1-羧酸 66016-28-2 详细
trans-4-{5-bromo-2-chloro-7H-pyrrolo[2,3-d]pyrimidin-7-yl}cyclohexan-1-ol 反式-4-{5-溴-2-氯-7H-吡咯并[2,3-d]嘧啶-7-基}环己-1-醇 1630906-40-9 详细
ethyl 2-(3-pyridylmethyl)pyrazole-3-carboxylate ethyl 1-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxylate 2250241-82-6 详细
(4R)-4-phenyl-1,3-oxazolidin-2-one (4R)-4-苯基-1,3-噁唑烷-2-酮 90319-52-1 详细
5-(2,2-difluorocyclopropyl)-1H-pyrazol-3-amine 5-(2,2-DIFLUOROCYCLOPROPYL)-1H-PYRAZOL-3-AMINE 1186609-07-3 详细
methyl 4-[2-(4-methoxyphenyl)-2-oxoethyl]benzoate 1416017-79-2 详细
1H,1'H-2,2'-biimidazole 联咪唑 492-98-8 详细
tert-butyl 3-cyclopropyl-3-hydroxy-azetidine-1-carboxylate 叔-丁基 3-环丙基-3-羟基吖丁啶-1-甲酸基酯 1438858-75-3 详细
2-[2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy]-4-methyl-pyrimidine 2-(2-氟-4-(4,4,5,5-四甲基-1,3,2-二氧硼杂环戊烷-2-基)苯氧基)-4-甲基嘧啶 2549188-28-3 详细
1-(4-bromopyrazol-1-yl)cyclopropanecarboxylic acid 1935387-65-7 详细
benzyl (2S)-2-{8-amino-1-bromoimidazo[1,5-a]pyrazin-3-yl}pyrrolidine-1-carboxylate 苯甲基 (2S)-2-{8-氨基-1-溴咪唑并[1,5-a]吡嗪-3-基}吡咯烷-1-甲酸基酯 1420478-88-1 详细
6,6'-dimethyl 5,5'-dibromo-2H,2'H,3H,3'H-[1,1'-biindole]-6,6'-dicarboxylate 6,6'-二甲基 5,5'-二溴-2H,2'H,3H,3'H-[1,1'-联吲哚]-6,6'-二甲酸基酯 2007910-50-9 详细
4-(cyclopropanesulfonyl)aniline 4-(环丙磺酰)苯胺 1147558-13-1 详细
3-(benzenesulfonylmethylene)oxetane 3-[(苯磺酰)甲亚基]噁丁环烷 1221819-46-0 详细
3-(3,5-difluorophenyl)pyrrolidine;hydrochloride 3-(3,5-二氟苯基)吡咯烷盐酸盐 2135332-31-7 详细
methyl 2-fluoro-5-(3-oxocyclobutyl)benzoate 2130017-23-9 详细
4-(dimethylamino)-4-phenylcyclohexan-1-one 4-(二甲氨基)-4-苯基环己烷-1-酮 65619-20-7 详细
(Z)-(ethyl N-{[4-cyclohexyl-3-(trifluoromethyl)phenyl]methoxy}ethanecarboximidate) N-[[4-环己基-3-(三氟甲基)苯基]甲氧基]亚氨基乙酸乙酯 1418144-65-6 详细
1-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl] -cyclobutanecarbonitrile 1-(4-(4,4,5,5-四甲基-1,3,2-二氧杂硼烷-2-基)苯基)环丁烷甲腈 1245831-55-3 详细
ethyl 5-amino-1-(4-fluorophenyl)pyrazole-4-carboxylate 5-氨基-1-(4-氟苯)吡唑-4-羧酸乙酯 138907-68-3 详细
tert-butyl 4-(5-iodopyrimidin-2-yl)piperazine-1-carboxylate 4-(5-碘嘧啶-2-基)哌啶-1-甲酸叔丁酯 1027616-32-5 详细
N-{5-bromoimidazo[1,2-a]pyridin-2-yl}cyclopropanecarboxamide N-{5-溴咪唑并[1,2-a]吡啶-2-基}环丙甲酰胺 1973485-26-5 详细
2-cyclohexyl-2-(1,3-dioxoisoindolin-2-yl)acetic acid 1218299-30-9 详细
(3S)-1-(oxetan-3-yl)pyrrolidin-3-ol (3S)-1-(氧杂环丁烷-3-基)吡咯烷-3-醇 1375415-97-6 详细
tert-butyl [3,3'-biazetidine]-1-carboxylate hydrochloride 3,3'-二氮杂环丁烷] -1-甲酸叔丁酯盐酸盐 2007910-70-3 详细
trans-2-(6-bromopyridin-3-yl)cyclopropan-1-amine dihydrochloride (1S,2R)-rel-2-(6-溴吡啶-3-基)环丙烷-1-胺二盐酸 918305-74-5 详细
3-bromo-1-tetrahydropyran-4-yl-pyrrolo[2,3-c]pyridine 3-溴-1-(四氢-2H-吡喃-4-基)-6-氮杂吲哚 956003-68-2 详细
3-(3-bromophenyl)-3-hydroxycyclobutane-1-carboxylic acid 1824170-45-7 详细
3-piperazin-1-yl-1,2-benzothiazole 4-(1,2-苯并异噻唑-3-基)-1-哌嗪 87691-87-0 详细
1-[(diphenylmethylidene)amino]cyclopropane-1-carbonitrile 1-[(二苯甲基负离子烯)氨基]环丙烷-1-甲腈 89985-88-6 详细
3-chloro-4-(pyridin-2-ylmethoxy)aniline 3-氯-4-(吡啶-2-基甲氧基)苯胺 524955-09-7 详细
2-phenyloxolane 2-苯基噁戊环 16133-83-8 详细
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