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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
(4-cyclopropylphenyl)boronic acid 302333-80-8 详细
4-[(3R)-1-tert-butoxycarbonyl-3-piperidyl]benzoic acid 1217749-88-6 详细
4-phenyl-2,8-diazaspiro[4.5]decan-1-one hydrochloride 4-苯基-2,8-二氮杂螺[4.5]癸烷-1-酮盐酸 1198284-29-5 详细
3-[1-oxo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)isoindolin-2-yl]piperidine-2,6-dione 2291363-98-7 详细
4-bromo-1-(oxolan-3-yl)-1H-pyrazole 1040377-07-8 详细
4-phenylbicyclo[2.2.2]octane-1-carboxylic acid 953-69-5 详细
tert-butyl (3S)-3-[tert-butyl(dimethyl)silyl]oxy-6-oxazol-4-yl-azepane-1-carboxylate 2940933-83-3 详细
tert-butyl 5-bromo-2-oxo-spiro[indoline-3,4'-piperidine]-1'-carboxylate 叔-丁基 5-溴-2-氧亚基-1,2-二氢螺[吲哚并-3,4'-哌啶]-1'-甲酸基酯 873779-30-7 详细
tert-butyl 3-morpholin-3-ylazetidine-1-carboxylate 2065250-71-5 详细
(1S,3aS,3bS,5aR,9aR,9bS,11aS)-9a,11a-dimethyl-7-oxo-1,2,3,3a,3b,4,5,5a,6,9b,10,11-dodecahydroindeno[5,4-f]quinoline-1-carboxylic acid 4-氮杂-5a-雄甾烷-1-烯-3-酮-17b-羧酸 104239-97-6 详细
4-(3-bromophenyl)-6,8-dichloro-2-methyl-1,2,3,4-tetrahydroisoquinoline hydrochloride 4-(3-溴苯基)-6,8-二氯-2-甲基-1,2,3,4-四氢异喹啉盐酸 543739-81-7 详细
spiro[2,3,5,7-tetrahydro-1H-pyrrolizine-6,1'-cyclopropane]-8-ylmethanol 1788873-88-0 详细
4-(3,4,5-trifluorophenyl)pyrrolidin-2-one 1263774-97-5 详细
3-(1-tert-butoxycarbonylazetidin-3-yl)bicyclo[1.1.1]pentane-1-carboxylic acid 2227205-20-9 详细
1-(phenylsulfanyl)bicyclo[1.1.1]pentane 98585-81-0 详细
tert-butyl 3-oxospiro[benzofuran-2,4-piperidine]-1-carboxylate 1207163-87-8 详细
methyl (2S,3S,4S,5R,6S)-3,4,5-triacetoxy-6-[2-[3-(9H-fluoren-9-ylmethoxycarbonylamino)propanoylamino]-4-(hydroxymethyl)phenoxy]tetrahydropyran-2-carboxylate 894096-02-7 详细
oxetan-3-yl(phenyl)methanol 2813635-48-0 详细
benzyl 1,2-dihydrospiro[indole-3,4'-piperidine]-1'-carboxylate 苯甲基 1,2-二氢螺[吲哚并-3,4'-哌啶]-1'-甲酸基酯 167484-18-6 详细
6-chlorospiro[1,2-dihydropyrrolo[3,2-c]pyridine-3,1'-cyclopropane 1860866-12-1 详细
methyl 2-tetrahydropyran-4-yl-1H-imidazole-4-carboxylate 1250150-10-7 详细
benzyl 3-piperazin-1-ylazetidine-1-carboxylate;dihydrochloride 2819572-05-7 详细
4-(1-tert-butoxycarbonyl-3-piperidyl)benzoic acid 916421-44-8 详细
2-bromoethyl(diphenyl)sulfonium;trifluoromethanesulfonate 247129-85-7 详细
1-methyl-3-(5-methyl-1,3,4-thiadiazol-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-one 详细
tert-butyl 5-bromospiro[indoline-3,4'-piperidine]-1'-carboxylate 叔-丁基 5-溴-1,2-二氢螺[吲哚并-3,4'-哌啶]-1'-甲酸基酯 878167-55-6 详细
1,2-dihydrospiro[indole-3,4'-piperidine]-2-one; trifluoroacetic acid 1,2-二氢螺[吲哚并-3,4'-哌啶]-2-酮; 三氟乙酸 1956371-16-6 详细
methyl (2S,3S,4S,5R,6S)-3,4,5-triacetoxy-6-[2-amino-4-(hydroxymethyl)phenoxy]tetrahydropyran-2-carboxylate 229977-57-5 详细
4-[(4-tert-butoxycarbonyl-1,4-diazepan-1-yl)sulfonyl]benzoic acid 874838-70-7 详细
5-[(2S)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-amine 1895867-65-8 详细
(1S,2R)-2-phenylcyclopropane-1-carboxylic acid (1S,2R)-2-苯基环丙烷-1-羧酸 23020-18-0 详细
2-(4-tert-butoxycarbonyl-1,4-diazepan-1-yl)-2-(2-naphthyl)acetic acid 885275-74-1 详细
5-amino-1,2,4-dithiazole-3-thione 6846-35-1 详细
6-bromo-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one hydrochloride 1650548-73-4 详细
4-(4-fluorophenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridine 1170034-47-5 详细
(1S)-2-(benzenesulfonyl)-1-[(2S)-pyrrolidin-2-yl]ethanol 2379295-70-0 详细
tert-butyl 4-(4-bromobenzenesulfonyl)piperidine-1-carboxylate 叔-丁基 4-(4-溴苯磺酰)哌啶-1-甲酸基酯 226398-62-5 详细
(3-phenylpiperidin-2-yl)methanol 130944-00-2 详细
4,5-dichlorodithiazol-1-ium;chloride 75318-43-3 详细
tert-butyl N-[1-(4-bromophenyl)cyclobutyl]carbamate 1032350-06-3 详细
5-pyrrolidin-2-yloxazole;dihydrochloride 1864014-35-6 详细
8,9-diazatricyclo[4.3.0.02]nona-1(6),7-diene-7-carboxylic acid 1372560-52-5 详细
4-(hydroxymethyl)-5-methyl-1,3-dioxol-2-one 91526-18-0 详细
(E)-N,N-dimethyl-N'-(3-sulfanylidene-3H-1,2,4-dithiazol-5-yl)methanimidamide 1192027-04-5 详细
benzyl 4-bromo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-carboxylate 473737-34-7 详细
ethyl 5-[(4S)-2,2-dimethyltetrahydropyran-4-yl]-1H-indole-2-carboxylate 2212021-77-5 详细
7'-nitro-1',2'-dihydrospiro[cyclopropane-1,3'-indole 1697091-16-9 详细
3-(m-tolyl)oxetan-3-ol 1511615-03-4 详细
4-(4-aminophenyl)morpholin-3-one 4-(4-氨基苯基)吗啉-3-酮 438056-69-0 详细
tert-butyl 7-bromospiro[indoline-3,4-piperidine]-1-carboxylate 叔-丁基 7-溴-1,2-二氢螺[吲哚并-3,4'-哌啶]-1'-甲酸基酯 1128133-41-4 详细
3,4-dihydrospiro[1-benzopyran-2,4'-piperidine]-4-one hydrochloride 159635-39-9 详细
7-[allyl(methyl)amino]-3-(diallylamino)-5,5-dimethyl-benzo[b][1]benzosilin-10-one 1807857-25-5 详细
3-bromo-5-(morpholin-4-yl)-7H-thieno[3,2-b]pyran-7-one 3-溴-5-(吗啉-4-基)-7H-噻吩并[3,2-b]吡喃-7-酮 1174429-23-2 详细
tert-butyl N-[1-(4-cyanophenyl)cyclobutyl]carbamate 叔-丁基 N-[1-(4-氰基苯基)环丁基]氨基甲酯 1032349-97-5 详细
oxalic acid;N-(oxetan-3-yl)piperidin-4-amine 2307737-94-4 详细
3-(3-bromophenyl)cyclobutanecarboxylic acid 1512074-73-5 详细
methylamino phenothiazine-10-carboxylate;hydrochloride 934812-38-1 详细
3-(4-bromophenyl)azetidin-3-amine;dihydrochloride 1384264-75-8 详细
2-(4-tert-butoxycarbonyl-1,4-diazepan-1-yl)-2-(2-thienyl)acetic acid 834884-95-6 详细
3-azatricyclo[4.2.2.02]decan-4-one 14932-32-2 详细
(4S)-4-phenylpyrrolidin-2-one 62624-45-7 详细
1-tert-butoxycarbonylspiro[indoline-3,4-piperidine]-5-carboxylic acid 888222-12-6 详细
benzyl 6-bromo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-carboxylate 473737-32-5 详细
4,5-dihydro-6-oxime-imidazo[4,5,1-jk][1]benzazepine-2,6,7(1h)-trione 4,5-二氢-6-肟-咪唑并[4,5,1-jk][1]苯氮杂卓-2,6,7(1h)-三酮 92260-82-7 详细
(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethan-1-amine hydrochloride 1948273-01-5 详细
tert-butyl 4-(4-bromo-1H-pyrazol-1-yl)piperidine-1-carboxylate 877399-50-3 详细
3-pyrrolidin-1-ylbicyclo[1.1.1]pentan-1-amine dihydrochloride 2792201-01-3 详细
(4R)-4-[(4-hydroxyphenyl)methyl]oxazolidine-2,5-dione 183732-21-0 详细
methyl 2-(1-methylpyrazol-4-yl)pyrimidine-4-carboxylate 2891598-98-2 详细
tert-butyl 5'-acetyl-3'H-spiro[azetidine-3,1'-[2]benzofuran]-1-carboxylate 叔-丁基 5'-乙酰基-3'H-螺[吖丁啶并-3,1'-[2]苯并呋喃]-1-甲酸基酯 1398609-81-8 详细
6-(1-methylpyrazol-3-yl)pyrazolo[1,5-a]pyrazin-4-ol 2940954-01-6 详细
{1-[(tert-butoxy)carbonyl]piperidin-4-yl}methyl 4-fluoro-4-(hydroxymethyl)piperidine-1-carboxylate {1-[(叔-丁氧基)羰基]哌啶-4-基}甲基 4-氟-4-(羟甲基)哌啶-1-甲酸基酯 2173112-50-8 详细
3-[3-(tert-butylsulfinylamino)oxetan-3-yl]benzoic acid 2665662-99-5 详细
tert-butyl 3-(1,2,4-oxadiazol-3-yl)azepane-1-carboxylate 2940939-18-2 详细
3-fluoro-4-(morpholin-4-yl)aniline 3-氟-4-(4-吗啉基)-苯胺 93246-53-8 详细
4-(chloromethyl)-5-methyl-1,3-dioxol-2-one 80841-78-7 详细
7'-nitrospiro[cyclopropane-1,3'-indoline]-2'-one 83414-08-8 详细
1,2-dihydrospiro[indole-3,4'-piperidine]-2-one 1,2-二氢螺[吲哚并-3,4'-哌啶]-2-酮 252882-61-4 详细
tert-butyl spiro[indoline-3,4-piperidine]-1-carboxylate 叔-丁基 1,2-二氢螺[吲哚并-3,4'-哌啶]-1'-甲酸基酯 180465-84-3 详细
2-[4-(tert-butoxycarbonylamino)-1-piperidyl]-2-(3-thienyl)acetic acid 885275-49-0 详细
1-ethyl-3-(4-nitrophenyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazole 942920-11-8 详细
tert-butyl 5'-bromo-3'H-spiro[azetidine-3,1'-[2]benzofuran]-1-carboxylate 叔-丁基 5'-溴-3'H-螺[吖丁啶并-3,1'-[2]苯并呋喃]-1-甲酸基酯 1398609-80-7 详细
2H,3H,5H,6H,8H,9H-1,4,7,10-tetraoxacyclododeca[2,3-g]quinolin-15-ol 2H,3H,5H,6H,8H,9H-1,4,7,10-四氧杂环十二碳六烯并[2,3-g]喹啉-15-酚 1355620-88-0 详细
4-phenyl-1H-pyrazole 10199-68-5 详细
4-tert-butyl-5-(hydroxymethyl)-1,3-dioxol-2-one 188525-93-1 详细
tert-butyl 4-[(3-bromo-5-methyl-2-pyridyl)methyl]-4-cyano-piperidine-1-carboxylate 2940942-93-6 详细
8-chloro-3-oxatricyclo[7.3.1.0]trideca-1(13),5,7,9,11-pentaene-2,4-dione 8-氯-3-氧杂三环[7.3.1.0]十三碳-1(13),5,7,9,11-五烯-2,4-二酮 4053-08-1 详细
2-[4-bromo-3-(3-chloro-5-cyano-phenoxy)-2-fluoro-phenyl]acetic acid 1007572-07-7 详细
(15R)-5-[2-chloro-5-(ethoxymethyl)pyrimidin-4-yl]oxy-15-methyl-11-thia-6,14,17-triazatetracyclo[8.8.02.0121]octadeca-1(10),2(7),3,5,8,12(18)-hexaen-13-one 1887069-10-4 详细
3-[1-methyl-6-(4-piperidyl)indazol-3-yl]piperidine-2,6-dione;hydrochloride 2888604-15-5 详细
3-(2-pyridyl)azetidin-3-ol;dihydrochloride 1415564-55-4 详细
2-chloro-4-[trans-3-amino-2,2,4,4-tetramethylcyclobutoxy]benzonitrile 2-氯-4-[反-3-氨基-2,2,4,4-四甲基环丁氧基]苯甲腈 1818885-54-9 详细
4-(3-methoxyazetidin-1-yl)piperidine;dihydrochloride 1400759-50-3 详细
ethyl 4-fluoro-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoate 2169699-38-9 详细
4-{[(9S)-9-hydroxy-2-azatricyclo[9.4.0.03,]pentadeca-1(11),3,5,7,12,14-hexaene-2-carbonyl]amino}butanoic acid 4-{[(9S)-9-羟基-2-氮杂三环[9.4.0.03,?]十五碳-1(11),3,5,7,12,14-六烯-2-羰基]氨基}丁酸 1523530-65-5 详细
4,5-dimethyl-1,3-dioxol-2-one 37830-90-3 详细
9-bromo-2-iodo-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine 1282516-69-1 详细
4-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]-1λ-thiane-1,1-dione 4-[4-(四甲基-1,3,2-二噁硼戊环-2-基)-1H-吡唑-1-基]-1λ?-硫烷-1,1-二酮 1778666-13-9 详细
(2,5-dioxopyrrolidin-1-yl) 3-[2-[2-[2-[2-(2,5-dioxopyrrol-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]propanoate 1325208-25-0 详细
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