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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
tert-butyl 4-(6-bromo-3-pyridyl)piperazine-1-carboxylate 412348-27-7 详细
3-(1H-pyrazol-4-yl)bicyclo[1.1.1]pentan-1-amine dihydrochloride 详细
3-[5-(azetidine-1-carbonyl)pyrazin-2-yl]oxy-5-[(1R)-2-methoxy-1-methyl-ethoxy]-N-(5-methylpyrazin-2-yl)benzamide 919784-13-7 详细
4-phenoxyaniline 4-苯氧基苯胺 139-59-3 详细
2-(2,5-difluorophenyl)-4-nitro-benzoic acid 1261942-55-5 详细
2-bromo-6-cyclopropyl-pyridine 1086381-26-1 详细
(1R)-2-phenyl-1-[(1S,2S,6R,8S)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,]decan-4-yl]ethan-1-amine hydrochloride 178455-03-3 详细
1-tetrahydropyran-4-ylpiperazine;dihydrochloride 790223-65-3 详细
3,3-difluoro-1-(1H-triazol-5-yl)cyclobutanamine;hydrochloride 2193057-66-6 详细
benzyl N-[2-tert-butyl-5-[(2R,4R)-4-hydroxytetrahydrofuran-2-yl]pyrazol-3-yl]carbamate 2821785-82-2 详细
4-chloro-2-cyclopropyl-pyrimidine 1044771-74-5 详细
cis-tert-butyl 3-(4-fluorobenzoyl)cyclobytylcarbamate 顺-叔-丁基 3-(4-氟苯甲酰)cyclobytylcarbamate 1630907-38-8 详细
trans-1-tert-butoxycarbonyl-3-phenyl-piperidine-4-carboxylic acid 1068522-17-7 详细
N-{2-chloropyrrolo[2,1-f][1,2,4]triazin-4-yl}-5-cyclopropyl-1H-pyrazol-3-amine N-{2-氯吡咯并[2,1-f][1,2,4]三嗪-4-基}-5-环丙基-1H-吡唑-3-胺 918538-08-6 详细
tert-butyl 4-[5-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazol-1-yl]piperidine-1-carboxylate 1092563-67-1 详细
4-[(5-bromo-3-pyridyl)sulfonyl]morpholine 889676-35-1 详细
tert-butyl N-[(3S,5R,6S)-6-methyl-2-oxo-5-phenyl-3-piperidyl]carbamate 1426936-02-8 详细
3-fluoro-4-(morpholin-4-yl)benzonitrile 588708-64-9 详细
3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]aniline 3-甲氧基-4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]苯胺 1254058-34-8 详细
cis-2,6-dimethyl-4-({4-[(E)-2-(tetramethyl-1,3,2-dioxaborolan-2-yl)ethenyl]phenyl}methyl)morpholine 顺-2,6-二甲基-4-({4-[(E)-2-(四甲基-1,3,2-二噁硼戊环-2-基)乙烯基]苯基}甲基)吗啉 1247001-44-0 详细
(5-methyl-2-oxo-1,3-dioxol-4-yl)methyl (4-nitrophenyl) carbonate 173604-87-0 详细
benzyl trans-4-ethoxy-2-(4-methoxycarbonylphenyl)piperidine-1-carboxylate 2756090-53-4 详细
(R)-benzofuran-2-yl(cyclopropyl)methanamine 1213316-22-3 详细
tert-butyl (3R)-3-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxylate hydrochloride 详细
2-(3,4-dichlorophenyl)pyrrolidine 298690-82-1 详细
2-pyridazin-4-ylthiazole-4-carboxylic acid 955400-58-5 详细
5-[(1S,4S)-2-oxa-5-azabicyclo[2.2.1]heptan-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxylic acid 2434843-95-3 详细
1-(3-pyridyl)cyclopropanamine 503417-38-7 详细
(2R,3R)-3-phenyltetrahydrofuran-2-carboxylic acid 1932359-39-1 详细
tert-butyl N-(1-pyrrolidin-3-ylcyclopropyl)carbamate 叔-丁基 1-(吡咯烷-3-基)环丙基氨基甲酯 185693-07-6 详细
2-phenyl-4H-oxazol-5-one 1199-01-5 详细
3-(azetidin-3-yl)pyridine;dihydrochloride 1236791-61-9 详细
3-cyclohexyl-4-nitro-1H-pyrazole 1247187-59-2 详细
4-cyclopropyl-3-methyl-1H-pyrazole 2411636-32-1 详细
(3R)-3-(4,4-difluoro-1-piperidyl)-3-(4-hydroxyphenyl)-7-(trifluoromethyl)indolin-2-one 2768139-76-8 详细
2-(diphenylphosphorylmethyl)phenol 70127-50-3 详细
3,5-dimethyl-1-(oxetan-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazole 2144759-94-2 详细
(3S,5S)-3-cyclopropyl-5-methyl-2-oxo-pyrrolidine-3-carbonitrile 1462289-99-1 详细
4-(1-piperidyl)pyridine 2767-90-0 详细
2-(2,6-dioxo-3-piperidyl)-5-nitro-isoindoline-1,3-dione 55003-81-1 详细
3-(azetidin-3-yl)-1H-pyrazole;bis(2,2,2-trifluoroacetic acid) 2225147-07-7 详细
tert-butyl 2-(azetidin-3-yl)azetidine-1-carboxylate;hemi(oxalic acid) 2940955-08-6 详细
4-cyclopropylsulfonylbenzenesulfonyl chloride 1556223-20-1 详细
4-(1,3-dioxolan-2-yl)-1-(2-nitrophenyl)piperidine 1317882-64-6 详细
2-(4-phenoxyphenyl)-7-(4-piperidyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide 1633350-04-5 详细
4-cyclopropyl-1,3-thiazole-2-carbaldehyde 211942-97-1 详细
tert-butyl N-[(3S,5R)-5-methyl-1-(3-nitro-4-pyridyl)-3-piperidyl]carbamate 1405128-33-7 详细
1-(1H-pyrazol-3-yl)cyclopropyl]methanol 2228778-26-3 详细
8-acetyl-6-methyl-2-phenyl-chromen-4-one 201815-65-8 详细
5-methyl-2-phenyl-oxazole-4-carboxylic acid 18735-74-5 详细
azetidin-1-yl-(5-chloropyrazin-2-yl)methanone 915948-98-0 详细
3-(3-chlorophenyl)cyclobutanecarboxylic acid 1781632-91-4 详细
tert-butyl (3S)-3-(4-amino-1-piperidyl)pyrrolidine-1-carboxylate;dihydrochloride 2920179-04-8 详细
1-tert-butyl-3-[[5-chloro-3-(chloromethyl)-2-pyridyl]methyl]-3H-pyrrolo[2,3-b]pyridin-2-one 1455358-12-9 详细
1-bromo-4-[difluoro(phenyl)methyl]benzene 152241-12-8 详细
2-bromo-6-(3-methoxytetrahydrofuran-3-yl)-4-methyl-pyridine 2368946-06-7 详细
tert-butyl trans-4-(4-aminocyclohexyl)-3-oxo-piperazine-1-carboxylate 1059623-58-3 详细
4-(cyclopropoxy)piperidine;hydrochloride 1147110-64-2 详细
3-(3-pyridylmethyl)-8-azabicyclo[3.2.1]octane;dihydrochloride 2098134-02-0 详细
2-(1,4-diazepan-1-yl)-2-(2-thienyl)acetic acid 1251039-68-5 详细
tert-butyl (4S)-4-(4-amino-1-piperidyl)-3,3-difluoro-piperidine-1-carboxylate 2891580-81-5 详细
trans-2-(3-fluorophenyl)cyclopropyl]methanamine hydrochloride 928054-07-3 详细
benzyl 4-[(3S)-4-tert-butoxycarbonyl-3-(cyanomethyl)piperazin-1-yl]-2-methylsulfanyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxylate 2206737-02-0 详细
4-bromo-1-(6-methoxy-3-pyridyl)indazole 1207478-79-2 详细
N,N'-bis(2-furylmethyl)oxamide 69010-90-8 详细
(2S,4R)-1-[(2S)-2-[6-[[2-[2,3-difluoro-6-(2-morpholinothiazol-4-yl)phenoxy]acetyl]amino]hexanoylamino]-3,3-dimethyl-butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methylthiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide 2488296-78-0 详细
tert-butyl (2S)-2-(4-bromophenyl)morpholine-4-carboxylate 1131220-37-5 详细
3-(5-bromo-3-methyl-2-oxo-benzimidazol-1-yl)piperidine-2,6-dione 2300099-98-1 详细
2-(3-bromo-4-methyl-phenyl)morpholine 1508643-74-0 详细
3-(5,6-difluoro-1-oxo-isoindolin-2-yl)piperidine-2,6-dione 2438241-40-6 详细
5-ethyl-2-fluoro-4-[4-fluoro-3-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)-1H-indazol-6-yl]phenol;dihydrochloride 2247925-44-4 详细
6-[[2-chloro-4-(trifluoromethyl)phenoxy]methyl]-5-ethyl-pyridine-2-carboxylic acid 2940957-33-3 详细
4-cyclopropoxybenzoic acid 62577-90-6 详细
3-(4-hydroxyphenyl)-3-(3,3,4,4-tetrafluoropyrrolidin-1-yl)-7-(trifluoromethyl)indolin-2-one 2768139-75-7 详细
N1-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]benzene-1,4-diamine 2261021-67-2 详细
trans-tert-butyl-dimethyl-[4-[5-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazol-1-yl]cyclohexoxy]silane 1350324-24-1 详细
(3S)-1-(4-piperidyl)piperidin-3-ol 1335117-24-2 详细
benzyl trans-4-[tert-butyl(diphenyl)silyl]oxy-2-(4-methoxycarbonylphenyl)piperidine-1-carboxylate 2751958-58-2 详细
2-chloro-5-[(4-isopropylphenyl)methylamino]phenyl]methanol 2940956-38-5 详细
4-[(pyridine-3-carbonylamino)methyl]benzoic acid 110576-10-8 详细
3-(oxetan-3-yl)-2-oxo-pyrrolidine-3-carbonitrile 1462289-86-6 详细
3-cyclopropyl-2-oxo-pyrrolidine-3-carbonitrile 1462287-25-7 详细
N-(p-tolyl)pyridin-3-amine 285991-95-9 详细
2-(2,6-dioxo-3-piperidyl)-5-ethynyl-isoindoline-1,3-dione 2154356-63-3 详细
3-(5-aminobenzofuran-3-yl)piperidine-2,6-dione 2618349-23-6 详细
7-chloro-8-fluoro-2-[[(2R,8S)-2-fluoro-1,2,3,5,6,7-hexahydropyrrolizin-8-yl]methoxy]-4-(2,2,2-trifluoroethoxy)pyrido[4,3-d]pyrimidine 2791271-54-8 详细
4,6-dichloro-2-(pyridin-3-yl)pyrimidine 4,6-二氯-2-(吡啶-3-基)嘧啶 89508-47-4 详细
5-(4-fluorophenyl)-2-methyl-4-(4-pyridyl)-1H-pyrimidin-6-one 208652-74-8 详细
5-(3-methoxy-4-pyridyl)pyrrolidin-3-ol;dihydrochloride 2940940-69-0 详细
methyl 2-(chloromethyl)-3-[[(2R)-oxetan-2-yl]methyl]benzimidazole-5-carboxylate 2436737-09-4 详细
(3R,4S)-1-(4-aminopyrimidin-2-yl)-3-fluoro-3-methyl-piperidin-4-ol 2660253-93-8 详细
(2R,5S)-5-benzylpiperidine-2-carboxylic acid 1221793-44-7 详细
3-tetrahydropyran-4-yloxyazetidine;hydrochloride 2098045-25-9 详细
2-bromo-6-[(3S)-3-methoxytetrahydrofuran-3-yl]-4-methyl-pyridine 2368946-04-5 详细
2-methyl-2-(4-oxetan-3-yl-piperazin-1-yl)-propionaldehyde 2-甲基-2-(4-氧杂环丁-3-基-哌嗪-1-基)丙醛 1575591-71-7 详细
1-(oxetan-3-yl)-1H-pyrazole-4-carboxylic acid 1389323-51-6 详细
hemi(oxalic acid) 3-phenylazetidine 2752460-78-7 详细
tert-butyl 2-(benzhydrylideneamino)acetate 81477-94-3 详细
5-[(pyrrolidin-1-yl)methyl]thiophene-2-carboxylic acid 733784-27-5 详细
2-(2,6-dioxo-3-piperidyl)-3-oxo-isoindoline-5-carboxylic acid 2171519-15-4 详细
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