N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide
![N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide price.](/CAS/GIF/702675-74-9.gif)
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- $28 - $5180
- Product name: N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide
- CAS: 702675-74-9
- MF: C23H26IN7O2S
- MW: 591.47
- EINECS:200-256-5
- MDL Number:MFCD12546134
- Synonyms:N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide;BX 795;N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)aMino]propyl]aMino]-2-pyriMidinyl]aMino]phenyl]-1-pyrrolidin;BX795/BX-795;N-(3-(5-IODO-4-(3-(THIOPHENE-2-CARBOXAMIDO)PROPYLAMINO)PYRIMIDIN-2-YLAMINO)PHENYL)PYRROLIDINE-1-CARBOXAMIDE;N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide BX-795;BX-795 hydrochloride;N-[3-[[5-iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-Pyrrolidinecarboxamide hydrochloride
45 prices
Selected condition：
Brand
- Adipogen Life Sciences
- AK Scientific
- Ambeed
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Axon Medchem
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- DC Chemicals
- Matrix Scientific
- Sigma-Aldrich
- Tocris
- TRC
- Usbiological
Package
- 2mg
- 10
- 1unit
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 200mg
- 250mg
- 50
- 1g
- 10mM(in 1mL DMSO)
- 1000mg
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1026-M005
- Product descriptionBX-795 ≥95%
- Packaging5mg
- Price$108
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number2292AH
- Product descriptionN-(3-(4-(2-(2-Formamidothiophen-3-yl)propanamido)-5-iodopyrimidin-2-ylamino)phenyl)pyrrolidine-1-carboxamide
- Packaging10mg
- Price$190
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number2292AH
- Product descriptionN-(3-(4-(2-(2-Formamidothiophen-3-yl)propanamido)-5-iodopyrimidin-2-ylamino)phenyl)pyrrolidine-1-carboxamide
- Packaging100mg
- Price$712
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA700044
- Product descriptionN-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+%
- Packaging5mg
- Price$46
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA700044
- Product descriptionN-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+%
- Packaging10mg
- Price$85
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA700044
- Product descriptionN-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+%
- Packaging25mg
- Price$184
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA700044
- Product descriptionN-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+%
- Packaging50mg
- Price$284
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA700044
- Product descriptionN-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+%
- Packaging100mg
- Price$436
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA700044
- Product descriptionN-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+%
- Packaging250mg
- Price$654
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA700044
- Product descriptionN-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+%
- Packaging1g
- Price$1633
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0000290
- Product descriptionBX 795 95.00%
- Packaging5MG
- Price$328.9
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8222
- Product descriptionBX-795
- Packaging1unit
- Price$28
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8222
- Product descriptionBX-795
- Packaging5mg
- Price$60
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8222
- Product descriptionBX-795
- Packaging10mM(in 1mL DMSO)
- Price$85
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8222
- Product descriptionBX-795
- Packaging10mg
- Price$110
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA8222
- Product descriptionBX-795
- Packaging50mg
- Price$380
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Adipogen Life Sciences | SYN-1026-M005 | BX-795 ≥95% | 5mg | $108 | 2021-12-16 | Buy |
| AK Scientific | 2292AH | N-(3-(4-(2-(2-Formamidothiophen-3-yl)propanamido)-5-iodopyrimidin-2-ylamino)phenyl)pyrrolidine-1-carboxamide | 10mg | $190 | 2021-12-16 | Buy |
| AK Scientific | 2292AH | N-(3-(4-(2-(2-Formamidothiophen-3-yl)propanamido)-5-iodopyrimidin-2-ylamino)phenyl)pyrrolidine-1-carboxamide | 100mg | $712 | 2021-12-16 | Buy |
| Ambeed | A700044 | N-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+% | 5mg | $46 | 2021-12-16 | Buy |
| Ambeed | A700044 | N-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+% | 10mg | $85 | 2021-12-16 | Buy |
| Ambeed | A700044 | N-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+% | 25mg | $184 | 2021-12-16 | Buy |
| Ambeed | A700044 | N-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+% | 50mg | $284 | 2021-12-16 | Buy |
| Ambeed | A700044 | N-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+% | 100mg | $436 | 2021-12-16 | Buy |
| Ambeed | A700044 | N-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+% | 250mg | $654 | 2021-12-16 | Buy |
| Ambeed | A700044 | N-(3-((5-Iodo-4-((3-(thiophene-2-carboxamido)propyl)amino)pyrimidin-2-yl)amino)phenyl)pyrrolidine-1-carboxamide 99+% | 1g | $1633 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0000290 | BX 795 95.00% | 5MG | $328.9 | 2021-12-16 | Buy |
| ApexBio Technology | A8222 | BX-795 | 1unit | $28 | 2021-12-16 | Buy |
| ApexBio Technology | A8222 | BX-795 | 5mg | $60 | 2021-12-16 | Buy |
| ApexBio Technology | A8222 | BX-795 | 10mM(in 1mL DMSO) | $85 | 2021-12-16 | Buy |
| ApexBio Technology | A8222 | BX-795 | 10mg | $110 | 2021-12-16 | Buy |
| ApexBio Technology | A8222 | BX-795 | 50mg | $380 | 2021-12-16 | Buy |
Properties
Melting point :>163°C (dec.)
Density :1.644
storage temp. :2-8°C
solubility :DMSO: soluble15mg/mL, clear
form :powder
pka :12.57±0.70(Predicted)
color :white to light brown
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
InChIKey :VAVXGGRQQJZYBL-UHFFFAOYSA-N
Density :1.644
storage temp. :2-8°C
solubility :DMSO: soluble15mg/mL, clear
form :powder
pka :12.57±0.70(Predicted)
color :white to light brown
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
InChIKey :VAVXGGRQQJZYBL-UHFFFAOYSA-N
Safety Information
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Description
3-Phosphoinositide-dependent protein kinase 1 (PDK1) is a serine-threonine kinase that phosphorylates and activates a range of other kinases, including PKB, PKA, and certain isoforms of PKC. BX-795 is a potent, ATP-competitive inhibitor of PDK1 in vitro (IC50 = 11 nM) and in cells (IC50 = 300 nM). At comparable concentrations, BX-795 also inhibits ERK8, MAPK-interacting kinase 2, Aurora B, Aurora C, MAP/microtubule affinity-regulating kinases 1-4, TNF receptor associated factor-associated NF-κB activator-binding kinase 1, IκB kinase ε, and additional kinases.Related product price
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![N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide](https://img.chemicalbook.com/ProductImageEN/2018-12/small/fe498182-1055-4d7c-bbd5-8bbb37f80631.png){kind=small}