Azilsartan
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- $5 - $2096
- Product name: Azilsartan
- CAS: 147403-03-0
- MF: C25H20N4O5
- MW: 456.45
- EINECS:808-058-6
- MDL Number:MFCD20278186
- Synonyms:AZILSARTAN;2-Ethoxy-1-[[2'-(4,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]methyl]benzimidazole-7-carboxylic acid Azilsartan;2-ethoxy -1- {[2'-(5-oxo-4,5-dihydro -1,2,4 -oxadiazol-3-yl) biphenyl-4-yl ] methyl} -1H –benzimi[d]dazole-7-carboxylic acid;2-ethoxy-1-((2'-(5-oxo-4,5-dihydro- 1,2,4-oxadiazol-3-yl)-[1,1'-biphenyl]-4-yl)methyl)-1H-benzo[d]imidazole-7-carboxylic acid;2-Ethoxy-1-[[2'-(4,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]methyl]benzimidazole-7-carboxylic acid;Tak 536;Unii-F9nux55p23;2-ethoxy-3-((2'-(5-oxo-2,5-dihydro-1,2,4-oxadiazol-3-yl)biphenyl-4-yl)Methyl)-3H-benzo[d]iMidazole-4-carboxylic acid
71 prices
Selected condition:
Brand
- aablocks
- AccelPharmtech
- ACHEMBLOCK
- AK Scientific
- Ambeed
- American Custom Chemicals Corporation
- ApexBio Technology
- AvaChem
- Axon Medchem
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- Chemcia Scientific
- Chem-Impex
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Matrix Scientific
- Sigma-Aldrich
- TCI Chemical
- Tocris
- TRC
- Usbiological
Package
- 10mM(in 1mL DMSO)
- 5mg
- 10mg
- 10mM(in1mLDMSO)
- 1MG
- 10
- 50
- 25mg
- 50mg
- 100mg
- 200MG
- 250mg
- 500mg
- 1.00g
- 1g
- 2g
- 5g
- 10g
- 25g
- 50g
- 100G
- Manufactureraablocks
- Product numberAA001ET2
- Product description1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98%
- Packaging10mg
- Price$8
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001ET2
- Product description1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98%
- Packaging100mg
- Price$12
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001ET2
- Product description1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98%
- Packaging250mg
- Price$15
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001ET2
- Product description1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98%
- Packaging1g
- Price$18
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001ET2
- Product description1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid ≥98%
- Packaging5g
- Price$70
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001ET2
- Product description1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98%
- Packaging25g
- Price$269
- Updated2026-05-28
- Buy
- ManufacturerAccelPharmtech
- Product numberLF1011
- Product descriptionAzilsartan 99.00%
- Packaging1G
- Price$280
- Updated2026-05-21
- Buy
- ManufacturerACHEMBLOCK
- Product numberF-4382
- Product descriptionAzilsartan 96%
- Packaging25G
- Price$240
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberF-4382
- Product descriptionAzilsartan 96%
- Packaging100G
- Price$605
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product numberB671
- Product descriptionAzilsartan
- Packaging5g
- Price$367
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product numberB671
- Product descriptionAzilsartan
- Packaging10g
- Price$401
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product numberJ11584
- Product descriptionAzilsartan
- Packaging5mg
- Price$30
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA217890
- Product descriptionAzilsartan 98+%
- Packaging1g
- Price$26
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA217890
- Product descriptionAzilsartan 98+%
- Packaging250mg
- Price$11
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA217890
- Product descriptionAzilsartan 98+%
- Packaging50mg
- Price$5
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA217890
- Product descriptionAzilsartan 98+%
- Packaging100mg
- Price$7
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA001ET2 | 1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98% | 10mg | $8 | 2026-05-28 | Buy |
| aablocks | AA001ET2 | 1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98% | 100mg | $12 | 2026-05-28 | Buy |
| aablocks | AA001ET2 | 1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98% | 250mg | $15 | 2026-05-28 | Buy |
| aablocks | AA001ET2 | 1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98% | 1g | $18 | 2026-05-28 | Buy |
| aablocks | AA001ET2 | 1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid ≥98% | 5g | $70 | 2026-05-28 | Buy |
| aablocks | AA001ET2 | 1-[[2'-(2,5-Dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl]-2-ethoxy-1H-benzimidazole-7-carboxylic acid 98% | 25g | $269 | 2026-05-28 | Buy |
| AccelPharmtech | LF1011 | Azilsartan 99.00% | 1G | $280 | 2026-05-21 | Buy |
| ACHEMBLOCK | F-4382 | Azilsartan 96% | 25G | $240 | 2026-05-27 | Buy |
| ACHEMBLOCK | F-4382 | Azilsartan 96% | 100G | $605 | 2026-05-27 | Buy |
| AK Scientific | B671 | Azilsartan | 5g | $367 | 2021-12-16 | Buy |
| AK Scientific | B671 | Azilsartan | 10g | $401 | 2021-12-16 | Buy |
| AK Scientific | J11584 | Azilsartan | 5mg | $30 | 2021-12-16 | Buy |
| Ambeed | A217890 | Azilsartan 98+% | 1g | $26 | 2021-12-16 | Buy |
| Ambeed | A217890 | Azilsartan 98+% | 250mg | $11 | 2021-12-16 | Buy |
| Ambeed | A217890 | Azilsartan 98+% | 50mg | $5 | 2021-12-16 | Buy |
| Ambeed | A217890 | Azilsartan 98+% | 100mg | $7 | 2021-12-16 | Buy |
Properties
Melting point :188 °C(dec.)
Density :1.42
storage temp. :Sealed in dry,2-8°C
solubility :DMSO: soluble15mg/mL (clear solution)
form :powder
pka :2.05±0.10(Predicted)
color :white to beige
InChIKey :KGSXMPPBFPAXLY-UHFFFAOYSA-N
SMILES :C1(OCC)N(CC2=CC=C(C3=CC=CC=C3C3=NC(=O)ON3)C=C2)C2=C(C(O)=O)C=CC=C2N=1
Density :1.42
storage temp. :Sealed in dry,2-8°C
solubility :DMSO: soluble15mg/mL (clear solution)
form :powder
pka :2.05±0.10(Predicted)
color :white to beige
InChIKey :KGSXMPPBFPAXLY-UHFFFAOYSA-N
SMILES :C1(OCC)N(CC2=CC=C(C3=CC=CC=C3C3=NC(=O)ON3)C=C2)C2=C(C(O)=O)C=CC=C2N=1
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||
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Description
Azilsartan is an antagonist of the angiotensin II type 1 receptor (AT1; IC50 = 0.42 μM) and the active metabolite of azilsartan medoxomil . Azilsartan is formed from azilsartan medoxomil by hydrolysis in the gastrointestinal tract and liver. Azilsartan also acts as an inverse agonist, inhibiting angiotensin II-induced accumulation of inositol-1-phosphate in COS-7 cells expressing recombinant human AT1 (IC50 = 2.6 nM). It reduces the maximal contractile response induced by angiotensin II in isolated rabbit aortic strips (pD2 = 9.9). Azilsartan (100 ng/kg, i.v.) inhibits the angiotensin II-induced pressor response in conscious normotensive rats.More related product prices
Aspartame Bifonazole Kresoxim-methyl Biphenyl Methyl salicylate Tribenuron methyl Tolvaptan 1H-BenziMidazole-7-carboxylic acid, 1-[[2'-(2,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]Methyl] -2-ethoxy-, ethyl ester O-Desethyl Azilsartan Azilsartan Medoxomil 4-(hidroximetil)-5-metil-1,3-dioxol-2-ona Methyl bromide 613-92-3Related product price
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Aspartame
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Bifonazole
$5-1403.6 -
Kresoxim-methyl
$24-1115
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