Filgotinib
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- $13 - $7020
- Product name: Filgotinib
- CAS: 1206161-97-8
- MF: C21H23N5O3S
- MW: 425.5
- EINECS:
- MDL Number:MFCD20527867
- Synonyms:SYN1158;CyclopropanecarboxaMide, N-[5-[4-[(1,1-dioxido-4-thioMorpholinyl)Methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]-;GLPG0634 (analog);N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide;N-(5-(4-((1,1-Dioxidothiomorpholino)methyl)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide;Filgotinib (GLPG0634);N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide Filgotinib (GLPG0634);GLPG0634(filgotinib)
78 prices
Selected condition：
Brand
- aablocks
- Abosyn
- ACHEMBLOCK
- Adipogen Life Sciences
- AK Scientific
- ApexBio Technology
- Apolloscientific
- Arctom
- AvaChem
- Biosynth
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- Matrix Scientific
- Medical Isotopes, Inc.
- Synthonix
- TRC
Package
- 10mM*1mLinDMSO(Solid+Solvent)
- 500mg
- 10mM(in1mLDMSO)
- 10mM*1mLinDMSO(Solution)
- 10mM*1mLinDMSO
- 100.00mg
- 250.00mg
- 1.00g
- 10g
- 10mM(in 1mL DMSO)
- 1mg
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- 5G
- Manufactureraablocks
- Product numberAA0039CS
- Product descriptionN-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99%
- Packaging1mg
- Price$13
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039CS
- Product descriptionN-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99%
- Packaging5mg
- Price$18
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039CS
- Product descriptionN-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99%
- Packaging10mg
- Price$22
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039CS
- Product descriptionN-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99%
- Packaging25mg
- Price$27
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039CS
- Product descriptionN-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99%
- Packaging50mg
- Price$37
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039CS
- Product descriptionN-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99%
- Packaging100mg
- Price$57
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039CS
- Product descriptionN-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99%
- Packaging250mg
- Price$112
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0039CS
- Product descriptionN-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide ≥98%
- Packaging1g
- Price$322
- Updated2026-05-28
- Buy
- ManufacturerAbosyn
- Product number61-11716
- Product descriptionN-(5-(4-((1,1-Dioxidothiomorpholino)methyl)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide 95-98%
- Packaging1g
- Price$270
- Updated2021-12-16
- Buy
- ManufacturerACHEMBLOCK
- Product numberI-9794
- Product descriptionFilgotinib 98%
- Packaging5G
- Price$340
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberI-9794
- Product descriptionFilgotinib 98%
- Packaging1G
- Price$80
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberI-9794
- Product descriptionFilgotinib 98%
- Packaging100MG
- Price$30
- Updated2026-05-27
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1158-M005
- Product descriptionGLPG0634 ≥95%
- Packaging5mg
- Price$346
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1158-M010
- Product descriptionGLPG0634 ≥95%
- Packaging10mg
- Price$497
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1158-M001
- Product descriptionGLPG0634 ≥95%
- Packaging1mg
- Price$205
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberSYN-1158-M050
- Product descriptionGLPG0634 ≥95%
- Packaging50mg
- Price$1415
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA0039CS | N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99% | 1mg | $13 | 2026-05-28 | Buy |
| aablocks | AA0039CS | N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99% | 5mg | $18 | 2026-05-28 | Buy |
| aablocks | AA0039CS | N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99% | 10mg | $22 | 2026-05-28 | Buy |
| aablocks | AA0039CS | N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99% | 25mg | $27 | 2026-05-28 | Buy |
| aablocks | AA0039CS | N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99% | 50mg | $37 | 2026-05-28 | Buy |
| aablocks | AA0039CS | N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99% | 100mg | $57 | 2026-05-28 | Buy |
| aablocks | AA0039CS | N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 99% | 250mg | $112 | 2026-05-28 | Buy |
| aablocks | AA0039CS | N-[5-[4-[(1,1-Dioxido-4-thiomorpholinyl)methyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide ≥98% | 1g | $322 | 2026-05-28 | Buy |
| Abosyn | 61-11716 | N-(5-(4-((1,1-Dioxidothiomorpholino)methyl)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide 95-98% | 1g | $270 | 2021-12-16 | Buy |
| ACHEMBLOCK | I-9794 | Filgotinib 98% | 5G | $340 | 2026-05-27 | Buy |
| ACHEMBLOCK | I-9794 | Filgotinib 98% | 1G | $80 | 2026-05-27 | Buy |
| ACHEMBLOCK | I-9794 | Filgotinib 98% | 100MG | $30 | 2026-05-27 | Buy |
| Adipogen Life Sciences | SYN-1158-M005 | GLPG0634 ≥95% | 5mg | $346 | 2026-05-06 | Buy |
| Adipogen Life Sciences | SYN-1158-M010 | GLPG0634 ≥95% | 10mg | $497 | 2026-05-06 | Buy |
| Adipogen Life Sciences | SYN-1158-M001 | GLPG0634 ≥95% | 1mg | $205 | 2026-05-06 | Buy |
| Adipogen Life Sciences | SYN-1158-M050 | GLPG0634 ≥95% | 50mg | $1415 | 2021-12-16 | Buy |
Properties
Melting point :229 - 231°C
Density :1.51±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :Soluble in DMSO (15 mg/ml with warming)
form :solid
pka :8.04±0.20(Predicted)
color :Off-white
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChI :InChI=1S/C21H23N5O3S/c27-20(17-8-9-17)23-21-22-19-3-1-2-18(26(19)24-21)16-6-4-15(5-7-16)14-25-10-12-30(28,29)13-11-25/h1-7,17H,8-14H2,(H,23,24,27)
InChIKey :RIJLVEAXPNLDTC-UHFFFAOYSA-N
SMILES :C1(C(NC2N=C3N(N=2)C(C2=CC=C(CN4CCS(=O)(=O)CC4)C=C2)=CC=C3)=O)CC1
Density :1.51±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :Soluble in DMSO (15 mg/ml with warming)
form :solid
pka :8.04±0.20(Predicted)
color :Off-white
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChI :InChI=1S/C21H23N5O3S/c27-20(17-8-9-17)23-21-22-19-3-1-2-18(26(19)24-21)16-6-4-15(5-7-16)14-25-10-12-30(28,29)13-11-25/h1-7,17H,8-14H2,(H,23,24,27)
InChIKey :RIJLVEAXPNLDTC-UHFFFAOYSA-N
SMILES :C1(C(NC2N=C3N(N=2)C(C2=CC=C(CN4CCS(=O)(=O)CC4)C=C2)=CC=C3)=O)CC1
Safety Information
| Symbol(GHS): |
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| Signal word: | Warning | ||||||||||||||||||||||||||||
| Hazard statements: |
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| Precautionary statements: |
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Description
Filgotinib (GLPG0634) is a selective JAK1 inhibitor with IC50 of 10 nM, 28 nM, 810 nM, and 116 nM for JAK1, JAK2, JAK3, and TYK2, respectively. Phase 2.Related product price
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Suppliers and manufacturers
Shandong Juntai Pharmaceutical Co., LTD.
Wuhan HSN Pharmaresearch CO., LTD.
Nanjing Vcare PharmaTech Co., Ltd
RD International Technology Co., Limited
Shanghai Boyle Chemical Co., Ltd.
ZHIWE CHEMTECH CO LTD
Chembest Research Laboratories Limited
Anhui Lianchuang Biological Medicine Co.,Ltd
Jinan Trio PharmaTech Co., Ltd.
Dalian Meilun Biotech Co., Ltd.