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25947-14-2

1-Phthalazineacetic acid, 3,4-dihydro-4-oxo-, Methyl ester synthesis

4synthesis methods
-

Yield:25947-14-2 66%

Reaction Conditions:

with thionyl chloride at 75; for 6 h;

References:

Mammoliti, Oscar;Jansen, Koen;El Bkassiny, Sandy;Palisse, Adeline;Triballeau, Nicolas;Bucher, Denis;Allart, Brigitte;Jaunet, Alex;Tricarico, Giovanni;De Wachter, Maxim;Menet, Christel;Blanc, Javier;Letfus, Vatroslav;Rup?i?, Renata;?mehil, Mario;Poljak, Tanja;Coornaert, Beatrice;Sonck, Kathleen;Duys, Inge;Waeckel, Ludovic;Lecru, Lola;Marsais, Florence;Jagerschmidt, Catherine;Auberval, Marielle;Pujuguet, Philippe;Oste, Line;Borgonovi, Monica;Wakselman, Emanuelle;Christophe, Thierry;Houvenaghel, Nicolas;Jans, Mia;Heckmann, Bertrand;Sanière, Laurent;Brys, Reginald [Journal of Medicinal Chemistry,2021,vol. 64,# 19,p. 14557 - 14586]