| Identification | Back Directory | [Name]
CHIR 2279 | [CAS]
158198-45-9 | [Synonyms]
CHIR 2279
Glycinamide, N-[2-(4-hydroxyphenyl)ethyl]glycyl-N-[1,1'-biphenyl]-4-ylglycyl-N2-(2-phenylethyl)- (9CI) | [Molecular Formula]
C34H36N4O4 | [MOL File]
158198-45-9.mol | [Molecular Weight]
564.67 |
| Hazard Information | Back Directory | [Uses]
CHIR-2279 is a high-affinity ligand (Ki=5 nM) for the α1-adrenergic receptor and can be further studied as a drug lead compound[1]. | [IC 50]
α1-adrenergic receptor: 5 nM (Ki) | [References]
[1] Zuckermann, et al. Discovery of nanomolar ligands for 7-transmembrane G-protein-coupled receptors from a diverse N-(substituted) glycine peptoid library. Journal of medicinal chemistry 37.17 (1994): 2678-2685. DOI:10.1021/jm00043a007 |
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