| Identification | Back Directory | [Name]
PITOFENONE HCL | [CAS]
54063-52-4 | [Synonyms]
Pitofenone
PITOFENONE HCL
Pitofenone D10
Pitofenone-d4 (deuterated)
Pitofenone (base and/or unspecified salts)
Methyl 2-{4-[2-(1-piperidinyl)ethoxy]benzoyl}benzoate
2-[4-[2-(1-Piperidinyl)ethoxy]benzoyl]benzoic acid methyl ester
Benzoic acid, 2-[4-[2-(1-piperidinyl)ethoxy]benzoyl]-, methyl ester
PitofenoneQ: What is
Pitofenone Q: What is the CAS Number of
Pitofenone Q: What is the storage condition of
Pitofenone | [Molecular Formula]
C22H25NO4 | [MDL Number]
MFCD01661944 | [MOL File]
54063-52-4.mol | [Molecular Weight]
367.44 |
| Hazard Information | Back Directory | [Uses]
Pitofenone, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively[1][2]. | [Definition]
ChEBI: Pitofenone is a member of benzophenones. | [IC 50]
AChE | [References]
[1] Bal-Tembe S, et al. HL 752: a potent and long-acting antispasmodic agent. Bioorg Med Chem. 1997 Jul;5(7):1381-7. DOI:10.1016/s0968-0896(97)00067-9
[2] Punekar NS, et al. Acetylcholinesterase inhibition by pitofenone: a spasmolytic compound. Biotechnol Appl Biochem. 1991 Dec;14(3):378-82. PMID:1777122 |
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