| Identification | Back Directory | [Name]
4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONE | [CAS]
869802-44-8 | [Synonyms]
A-794282
4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONE
Pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(3H)-one, 9-(dimethylamino)-3-(4-ethylphenyl)- | [Molecular Formula]
C19H18N4OS | [MDL Number]
MFCD11501299 | [MOL File]
869802-44-8.mol | [Molecular Weight]
350.44 |
| Hazard Information | Back Directory | [Description]
A-794282 is a selective mGluR1 antagonist. | [Uses]
A-794282 is a compound with analgesic activity and is a selective mGlu1 receptor antagonist that significantly reduces pain behaviors in a postoperative pain model, but motor side effects may occur at higher doses. | [IC 50]
mGluR1 | [References]
[1] Analgesic activity of metabotropic glutamate receptor 1 antagonists on spontaneous post-operative pain in rats DOI:10.1016/j.ejphar.2007.09.047
[2] [Research progress of selective mGluR1 antagonists] PMID:22242445 |
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cjbscvictory
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13348960310 |
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https://www.weikeqi-biotech.com/ |
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