5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE

5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE structure

CAS No.: 144625-67-2

Chemical Name:: 5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE

Synonyms: GR 125487;GR 125487 SULFAMATE;GR 125487 SULFAMATE SALT;(1-(2-(Methylsulfonamido)ethyl)piperidin-4-yl)-methyl 5-fluoro-2-methoxy-1H-indole-3-carboxyla;(1-(2-(Methylsulfonamido)ethyl)piperidin-4-yl)-methyl 5-fluoro-2-methoxy-1H-indole-3-carboxylate;5-Fluoro-2-methoxy-[1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]-1H-indole-3-methylcarboxylatesulfamate;5-fluoro-2-Methoxy-1H-Indole-3-carboxylic acid-[1-[2-[(Methylsulfonyl)aMino]ethyl]-4-piperidinyl]Methyl ester;5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE;1H-Indole-3-carboxylic acid, 5-fluoro-2-methoxy-, [1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]methyl ester;[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]METHYL 5-FLUORO-2-METHOXY-1H-INDOLE-3-CARBOXYLATE SULFAMATE SALT

CBNumber:: CB2346616

Molecular Formula:: C19H26FN3O5S

Molecular Weight:: 427.49

MDL Number:: MFCD00912900

MOL File:: 144625-67-2.mol

MSDS File:: SDS

Last updated:2023-04-23 13:52:06

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5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE Properties

Melting point	118-120℃
Boiling point	613.4±65.0 °C(Predicted)
Density	1.313±0.06 g/cm3(Predicted)
storage temp.	Sealed in dry,2-8°C
solubility	H₂O: ~14 mg/mL at 60 °C, soluble
form	solid
pka	11.22±0.40(Predicted)
color	off-white

SAFETY

Risk and Safety Statements

WGK Germany	3

5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE price More Price(12)

Manufacturer	Product number	Product description	CAS number	Packaging	Price	Updated	Buy
Tocris	1658	GR125487sulfamate ≥97%(HPLC)	144625-67-2	10	$223	2021-12-16	Buy
Tocris	1658	GR125487sulfamate ≥97%(HPLC)	144625-67-2	50	$872	2021-12-16	Buy
Usbiological	451421	GR 125487 Sulfamate	144625-67-2	1mg	$389	2021-12-16	Buy
American Custom Chemicals Corporation	API0008782	5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE 95.00%	144625-67-2	10MG	$714.32	2021-12-16	Buy
AK Scientific	7131AA	(1-(2-(Methylsulfonamido)ethyl)piperidin-4-yl)methyl5-fluoro-2-methoxy-1H-indole-3-carboxylate	144625-67-2	250mg	$1051	2021-12-16	Buy

Product number	Packaging	Price	Buy
1658	10	$223	Buy
1658	50	$872	Buy
451421	1mg	$389	Buy
API0008782	10MG	$714.32	Buy
7131AA	250mg	$1051	Buy

5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE Chemical Properties,Uses,Production

Uses

GR 125487 Sulfamate is potent, selective 5-HT4 antagonist; active in vivo.

Biological Activity

Potent and selective 5-HT 4 receptor antagonist (K i = 0.19 nM for porcine 5-HT 4 ). Centrally active following systemic administration in vivo .

5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE Preparation Products And Raw materials

Raw materials

Preparation Products

5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE Suppliers

Global( 19)Suppliers

Supplier	Tel	Email	Country	ProdList	Advantage
Amadis Chemical Company Limited	571-89925085	sales@amadischem.com	China	131981	58
3B Pharmachem (Wuhan) International Co.,Ltd.	821-50328103-801 18930552037	3bsc@sina.com	China	15848	69
Jiangsu Aikon Biopharmaceutical R&D co.,Ltd.	025-66113011 18112977050	cb6@aikonchem.com	China	16687	50
EMMX Biotechnology LLC	888-539-0666	info@emmx.com	United States	8449	60
Shanghai Universal Biotech Co.,Ltd	18768175414	gaojun@univ-bio.com	China	24998	58

Supplier	Advantage
Amadis Chemical Company Limited	58
3B Pharmachem (Wuhan) International Co.,Ltd.	69
Jiangsu Aikon Biopharmaceutical R&D co.,Ltd.	50
EMMX Biotechnology LLC	60
Shanghai Universal Biotech Co.,Ltd	58

144625-67-2(5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE)Related Search:

5-FLUOROINDOLE-3-CARBOXYLIC ACID 5-FLUORO-1H-INDOLE-3-CARBOXYLIC ACID METHYL ESTER 5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE [1-(2-aminoethyl)-4-piperidinyl]methanol 5-FLUOROINDOLE-3-CARBOXALDEHYDE

[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]METHYL 5-FLUORO-2-METHOXY-1H-INDOLE-3-CARBOXYLATE SULFAMATE SALT 5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE GR 125487 SULFAMATE GR 125487 SULFAMATE SALT 5-Fluoro-2-methoxy-[1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]-1H-indole-3-methylcarboxylatesulfamate 5-fluoro-2-Methoxy-1H-Indole-3-carboxylic acid-[1-[2-[(Methylsulfonyl)aMino]ethyl]-4-piperidinyl]Methyl ester GR 125487 (1-(2-(Methylsulfonamido)ethyl)piperidin-4-yl)-methyl 5-fluoro-2-methoxy-1H-indole-3-carboxylate (1-(2-(Methylsulfonamido)ethyl)piperidin-4-yl)-methyl 5-fluoro-2-methoxy-1H-indole-3-carboxyla 1H-Indole-3-carboxylic acid, 5-fluoro-2-methoxy-, [1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]methyl ester 144625-67-2 C19H26FN3O5SSO3NH2 C19H26FN3O5SH2NSO3H C19H26FN3O5S