CAY10498
- CAS No.
- 863202-33-9
- Chemical Name:
- CAY10498
- Synonyms
- CAY10498;A3AR antagonist 3;CAY10498,CAY-10498;2-phenyl-amino-N6-endo-norbornyladenine;CAY10498, A3 adenosine receptor antagonist;6-N-(3-bicyclo[2.2.1]heptanyl)-2-N-phenyl-7H-purine-2,6-diamine;1H-Purine-2,6-diamine, N6-(1R,2S,4S)-bicyclo(2.2.1)hept-2-yl-N2-phenyl;9H-Purine-2,6-diamine, N6-(1R,2S,4S)-bicyclo[2.2.1]hept-2-yl-N2-phenyl-, rel-
- CBNumber:
- CB32590412
- Molecular Formula:
- C18H20N6
- Molecular Weight:
- 320.39
- MDL Number:
- MFCD23160216
- MOL File:
- 863202-33-9.mol
| Product description | Number | Pack Size | Price |
| CAY10498 ≥95% | 10007955 | 500μg | $121 |
| CAY10498 ≥95% | 10007955 | 1mg | $218 |
| CAY10498 ≥95% | 10007955 | 5mg | $961 |
| 1H-Purine-2,6-diamine,N6-(1R,2S,4S)-bicyclo(2.2.1)hept-2-yl-N2-phenyl | 1287AH | 5mg | $1169 |
| 1H-PURINE-2,6-DIAMINE, N6-(1R,2S,4S)-BICYCLO(2.2.1)HEPT-2-YL-N2-PHENYL 95.00% | NUC0002272 | 5MG | $502.99 |
CAY10498 price More Price(5)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Cayman Chemical | 10007955 | CAY10498 ≥95% | 863202-33-9 | 500μg | $121 | 2024-03-01 | Buy |
| Cayman Chemical | 10007955 | CAY10498 ≥95% | 863202-33-9 | 1mg | $218 | 2024-03-01 | Buy |
| Cayman Chemical | 10007955 | CAY10498 ≥95% | 863202-33-9 | 5mg | $961 | 2024-03-01 | Buy |
| AK Scientific | 1287AH | 1H-Purine-2,6-diamine,N6-(1R,2S,4S)-bicyclo(2.2.1)hept-2-yl-N2-phenyl | 863202-33-9 | 5mg | $1169 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | NUC0002272 | 1H-PURINE-2,6-DIAMINE, N6-(1R,2S,4S)-BICYCLO(2.2.1)HEPT-2-YL-N2-PHENYL 95.00% | 863202-33-9 | 5MG | $502.99 | 2021-12-16 | Buy |
CAY10498 Chemical Properties,Uses,Production
Uses
A3AR antagonist 3 (compound 21) is a selective A3 adenosine receptor (A3AR) antagonist with a Ki of 37 nM. A3AR antagonist 3 shows >60-fold selectivity in comparison to A1 and A2A adenosine receptors[1].
IC 50
hA3: 37 nM (Ki); hA1AR: 2.22 μM (Ki); hA2AAR: 7.73 μM (Ki)
References
[1] Melissa Perreira, et al. "Reversine" and its 2-substituted adenine derivatives as potent and selective A3 adenosine receptor antagonists. J Med Chem. 2005 Jul 28;48(15):4910-8. DOI:10.1021/jm050221l
CAY10498 Preparation Products And Raw materials
Raw materials
Preparation Products
CAY10498 Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| TargetMol Chemicals Inc. | +1-781-999-5354; +17819995354 | marketing@targetmol.com | United States | 32435 | 58 |
| Aladdin Scientific | tp@aladdinsci.com | United States | 52923 | 58 | |
| DAYANG CHEM (HANGZHOU) CO.,LTD | +86-88938639 +86-17705817739 | info@dycnchem.com | China | 53899 | 58 |
| BOC Sciences | 1-631-485-4226; 16314854226 | info@bocsci.com | United States | 12952 | 65 |
| BOC Sciences | 16314854226 | info@bocsci.com | United States | 9923 | 65 |
| Shanghai EFE Biological Technology Co., Ltd. | 021-65675885 18964387627 | info@efebio.com | China | 9803 | 58 |
| Shanghai Hongye Biotechnology Co. Ltd | 400-9205774 | sales@glpbio.cn | China | 6777 | 58 |
| ChemeGen(Shanghai) Biotechnology Co.,Ltd. | 18818260767 | sales@chemegen.com | China | 11218 | 58 |
| Taizhou Nanfeng Pharmaceutical Research Institute | nanfengdrug@163.com; 18616377689 | nanfengdrug@163.com | China | 20009 | 58 |
| TargetMol Chemicals Inc. | 4008200310 | marketing@tsbiochem.com | China | 24961 | 58 |





