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GI 254023X

GI 254023X Structure
GI 254023X structure
CAS No.
260264-93-5
Chemical Name:
GI 254023X
Synonyms
GI4023;GI 254023X;SRI 028594);GI 254023X(GI 4023;GI254023X[SML0789];GI254023X, 10 mM in DMSO;GI 254023X;GI-254023X;GI4023;SRI028594;GI254023X; GI 254023X; GI-254023X;GI4023; GI-4023; GI 4023;(R)-N-((S)-3,3-Dimethyl-1-(methylamino)-1-oxobutan-2-yl)-2-((S)-1-(N-hydroxyformamido)ethyl)-5-phenylpentanamide;(2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-2-[(1S)-1-(N-hydroxyformamido)ethyl]-5-phenylpentanamide
CBNumber:
CB82650737
Molecular Formula:
C21H33N3O4
Molecular Weight:
391.51
MDL Number:
MFCD19381832
MOL File:
260264-93-5.mol
MSDS File:
SDS
TDS File:
TDS
Last updated:2026-08-20 20:20:01
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GI 254023X Properties

Density 1.112±0.06 g/cm3(Predicted)
storage temp. 2-8°C
solubility DMSO: soluble15mg/mL, clear
pka 8.48±0.69(Predicted)
form powder
color white to beige
InChIKey GHVMTHKJUAOZJP-CGTJXYLNSA-N
SMILES ON(C=O)[C@@H](C)[C@@H](CCCC1=CC=CC=C1)C(N[C@@H](C(C)(C)C)C(NC)=O)=O
UNSPSC Code 12352200
NACRES NA.77

SAFETY

Risk and Safety Statements

WGK Germany  3
Storage Class 11 - Combustible Solids

GI 254023X price More Price(56)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Sigma-Aldrich SML0789 GI254023X ≥98% (HPLC) 260264-93-5 5mg $234 2026-04-30 Buy
Sigma-Aldrich SML0789 GI254023X ≥98% (HPLC) 260264-93-5 25mg $933 2026-04-30 Buy
Cayman Chemical 28284 GI 254023X ≥98% 260264-93-5 1mg $63 2026-04-30 Buy
Cayman Chemical 28284 GI 254023X ≥98% 260264-93-5 5mg $183 2026-04-30 Buy
Cayman Chemical 28284 GI 254023X ≥98% 260264-93-5 10mg $303 2026-04-30 Buy
Product number Packaging Price Buy
SML0789 5mg $234 Buy
SML0789 25mg $933 Buy
28284 1mg $63 Buy
28284 5mg $183 Buy
28284 10mg $303 Buy

GI 254023X Chemical Properties, Uses, Production

Uses

GI 254023X is an ADAM10 metaloproteinase inhibitor.

Uses

GI254023X has been used to inhibit ADAM10 (ADAM metallopeptidase domain 10).

Definition

ChEBI: GI254023X is a L-valine derivative that is 3-methyl-L-valine in which carboxy OH group is replaced by a methylnitrilo group and the one of the amino hydrogens is replaced by a (2R)-2-{(1S)-1-[formyl(hydroxy)amino]ethyl}-5-phenylpentanoyl group. It is a potent MMP9 and ADAM10 metalloprotease inhibitor with IC50 of 2.5 and 5.3 nM, respectively. It has a role as an apoptosis inducer, an antineoplastic agent, a matrix metalloproteinase inhibitor and an EC 3.4.24.* (metalloendopeptidase) inhibitor. It is a L-valine derivative, an aldehyde and a member of hydroxylamines.

Biochem/physiol Actions

GI254023X is a potent and selective ADAM10 metalloproteinase inhibitor.

storage

Store at -20°C

GI 254023X Preparation Products And Raw materials

Raw materials

Preparation Products

GI 254023X Suppliers

Global Suppliers ( 138)
Supplier Tel Email Country ProdList Advantage
Chembest Research Laboratories Limited 021-20908456 sales@BioChemBest.com China 5996 61
BOC Sciences 1-631-485-4226; 16314854226 info@bocsci.com United States 9920 65
Okeanos Tech Co,. Ltd. 010-62651721 18610486005 minghui.yu@okeanos.com.cn China 495 60
Shanghai Topbiochem Technology Co., Ltd 021-58170097 info@topbiochem.com China 9509 58
MedChemexpress LLC 021-58955995 sales@medchemexpress.cn United States 4853 58
Nanjing Dulai Biotechnology Co., Ltd. 025-84699383-8003;025-846993838003-8003 18013301590 njduly@126.com China 3293 55
AdooQ BioScience, LLC +1 (866) 930-6790 info@adooq.com United States 2774 58
TargetMol Chemicals Inc. 021-021-33632979 15002134094 marketing@targetmol.com China 7993 58
Bide Pharmatech Ltd. 400-164-7117 18317119277 product02@bidepharm.com China 40000 60
AdooQ Bioscience CHINA 025-58849295 info@adooq.cn China 2981 60
Supplier Advantage
Chembest Research Laboratories Limited 61
BOC Sciences 65
Okeanos Tech Co,. Ltd. 60
Shanghai Topbiochem Technology Co., Ltd 58
MedChemexpress LLC 58
Nanjing Dulai Biotechnology Co., Ltd. 55
AdooQ BioScience, LLC 58
TargetMol Chemicals Inc. 58
Bide Pharmatech Ltd. 60
AdooQ Bioscience CHINA 60

View Latest Price from GI 254023X manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
GI254023X pictures 2026-08-20 GI254023X
260264-93-5
 $97.00-198.00 98.55% 10g TargetMol Chemicals Inc.
GI 254023X pictures 2026-06-30 GI 254023X
260264-93-5
 1KG 98% 1000kg Shaanxi Dideu New Materials Co. Ltd
  • GI254023X pictures
  • GI254023X
    260264-93-5
  • $97.00-198.00
  • 98.55%
  • TargetMol Chemicals Inc.
  • GI 254023X pictures
  • GI 254023X
    260264-93-5
  • $0.00
  • 98%
  • Shaanxi Dideu New Materials Co. Ltd

GI 254023X Spectrum

GI 254023X(260264-93-5)1HNMR

260264-93-5 (GI 254023X) Related Search:

PRND Nr N,N-Dimethylcyclohexylamine (1S,2S)-N,N'-Dihydroxy-N,N'-bis(3,3,3-triphenylpropionyl)cyclohexane-1,2-diamine N-(R)-[2-(Hydroxyaminocarbonyl)methyl]-4-methylpentanoyl-L-naphthylalanyl-L-alanine amide
TAPI-0

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GI 254023X (2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]-propyl]-2-[(1S)-1-[formyl(hydroxy)amino]ethyl]-5-phenylpentanamide GI4023 GI 254023X(GI 4023 SRI 028594) GI 254023X;GI-254023X;GI4023;SRI028594 (2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-2-[(1S)-1-(N-hydroxyformamido)ethyl]-5-phenylpentanamide ((2R,3S)-3-(formyl-hydroxyamino)-2-(3-phenyl-1-propyl)butanoic acid [(1S)-2,2-dimethyl-1-methylcarbamoyl-1-propyl] amide) (alphaR)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-alpha-[(1S)-1-(formylhydroxyamino)ethyl]benzenepentanamide GI254023X; GI 254023X; GI-254023X;GI4023; GI-4023; GI 4023 Benzenepentanamide, N-[(1S)-2,2-dimethyl-1-[(methylamino)carbonyl]propyl]-α-[(1S)-1-(formylhydroxyamino)ethyl]-, (αR)- (R)-N-((S)-3,3-Dimethyl-1-(methylamino)-1-oxobutan-2-yl)-2-((S)-1-(N-hydroxyformamido)ethyl)-5-phenylpentanamide GI254023X, 10 mM in DMSO GI254023X[SML0789] 260264-93-5 GI 254023X