ChemicalBook >> CAS DataBase List >>GI 254023X
GI 254023X
- CAS No.
- 260264-93-5
- Chemical Name:
- GI 254023X
- Synonyms
- GI4023;GI 254023X;SRI 028594);GI 254023X(GI 4023;GI 254023X;GI-254023X;GI4023;SRI028594;GI254023X; GI 254023X; GI-254023X;GI4023; GI-4023; GI 4023;(R)-N-((S)-3,3-Dimethyl-1-(methylamino)-1-oxobutan-2-yl)-2-((S)-1-(N-hydroxyformamido)ethyl)-5-phenylpentanamide;(2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-2-[(1S)-1-(N-hydroxyformamido)ethyl]-5-phenylpentanamide;Benzenepentanamide, N-[(1S)-2,2-dimethyl-1-[(methylamino)carbonyl]propyl]-α-[(1S)-1-(formylhydroxyamino)ethyl]-, (αR)-;(2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]-propyl]-2-[(1S)-1-[formyl(hydroxy)amino]ethyl]-5-phenylpentanamide
- CBNumber:
- CB82650737
- Molecular Formula:
- C21H33N3O4
- Molecular Weight:
- 391.51
- MDL Number:
- MFCD19381832
- MOL File:
- 260264-93-5.mol
- MSDS File:
- SDS
Last updated:2023-06-30 15:45:59
GI 254023X price More Price(20)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich | SML0789 | GI254023X ≥98% (HPLC) | 260264-93-5 | 5mg | $212 | 2024-03-01 | Buy |
| Sigma-Aldrich | SML0789 | GI254023X ≥98% (HPLC) | 260264-93-5 | 25mg | $847 | 2024-03-01 | Buy |
| Cayman Chemical | 28284 | GI 254023X | 260264-93-5 | 1mg | $57 | 2024-03-01 | Buy |
| Cayman Chemical | 28284 | GI 254023X | 260264-93-5 | 25mg | $479 | 2024-03-01 | Buy |
| Cayman Chemical | 28284 | GI 254023X | 260264-93-5 | 5mg | $166 | 2024-03-01 | Buy |
GI 254023X Chemical Properties,Uses,Production
Uses
GI 254023X is an ADAM10 metaloproteinase inhibitor.
Uses
GI254023X has been used to inhibit ADAM10 (ADAM metallopeptidase domain 10).
Definition
ChEBI: GI254023X is a L-valine derivative that is 3-methyl-L-valine in which carboxy OH group is replaced by a methylnitrilo group and the one of the amino hydrogens is replaced by a (2R)-2-{(1S)-1-[formyl(hydroxy)amino]ethyl}-5-phenylpentanoyl group. It is a potent MMP9 and ADAM10 metalloprotease inhibitor with IC50 of 2.5 and 5.3 nM, respectively. It has a role as an apoptosis inducer, an antineoplastic agent, a matrix metalloproteinase inhibitor and an EC 3.4.24.* (metalloendopeptidase) inhibitor. It is a L-valine derivative, an aldehyde and a member of hydroxylamines.
Biochem/physiol Actions
GI254023X is a potent and selective ADAM10 metalloproteinase inhibitor.
storage
Store at -20°C
GI 254023X Preparation Products And Raw materials
Raw materials
Preparation Products
GI 254023X Suppliers
Global( 97)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Career Henan Chemica Co | +86-0371-86658258 15093356674; | laboratory@coreychem.com | China | 30255 | 58 |
| Hefei Hirisun Pharmatech Co., Ltd | +8615056975894 | shawn@hirisunpharm.com | CHINA | 9923 | 58 |
| Nextpeptide Inc | +86-0571-81612335 +8613336028439 | sales@nextpeptide.com | China | 19915 | 58 |
| InvivoChem | +1-708-310-1919 +1-13798911105 | sales@invivochem.cn | United States | 6393 | 58 |
| Nantong HI-FUTURE Biology Co., Ltd. | +undefined18051384581 | sales@chemhifuture.com | China | 3136 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354 | support@targetmol.com | United States | 19973 | 58 |
| Wuhan Topule Biopharmaceutical Co., Ltd | +8618327326525 | masar@topule.com | China | 8474 | 58 |
| Shenyang Zhongshen Zekang Biomedical Technology Research Co., Ltd | +86-18341751992 +86-15382112998 | 757984502@qq.com | China | 892 | 58 |
| Young Lively PharminBlock Co.,Ltd | +undefined18600731423 | jason_gao@yl-pharminblock.com | China | 1944 | 58 |
| Aladdin Scientific | +1-+1(833)-552-7181 | sales@aladdinsci.com | United States | 57511 | 58 |
260264-93-5(GI 254023X)Related Search:
GI 254023X
(2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]-propyl]-2-[(1S)-1-[formyl(hydroxy)amino]ethyl]-5-phenylpentanamide
GI4023
GI 254023X(GI 4023
SRI 028594)
GI 254023X;GI-254023X;GI4023;SRI028594
(2R)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-2-[(1S)-1-(N-hydroxyformamido)ethyl]-5-phenylpentanamide
((2R,3S)-3-(formyl-hydroxyamino)-2-(3-phenyl-1-propyl)butanoic acid [(1S)-2,2-dimethyl-1-methylcarbamoyl-1-propyl] amide)
(alphaR)-N-[(1S)-2,2-Dimethyl-1-[(methylamino)carbonyl]propyl]-alpha-[(1S)-1-(formylhydroxyamino)ethyl]benzenepentanamide
GI254023X; GI 254023X; GI-254023X;GI4023; GI-4023; GI 4023
Benzenepentanamide, N-[(1S)-2,2-dimethyl-1-[(methylamino)carbonyl]propyl]-α-[(1S)-1-(formylhydroxyamino)ethyl]-, (αR)-
(R)-N-((S)-3,3-Dimethyl-1-(methylamino)-1-oxobutan-2-yl)-2-((S)-1-(N-hydroxyformamido)ethyl)-5-phenylpentanamide
260264-93-5