プレドニゾロンリン酸エステルナトリウム 化学特性,用途語,生産方法
外観
白色~ほとんど白色粉末~結晶
効能
抗炎症薬, グルココルチコイド受容体作動薬
説明
Prednisolone is a synthetic analog of the natural glucocorticoid corticosterone that has anti-
inflammatory and immunsuppressive actions. It avidly binds both glucocorticoid and mineralocorticoid receptors (K
is = 2.4 and 37 nM). Prednisolone Phosphate, prepared as the sodium salt, is a water-
soluble ester of the poorly soluble parent molecule, prednisolone. It is rapidly hydrolyzed
in vivo to the parent molecule when administered intravenously. In addition, when given orally, prednisolone phosphate is more readily absorbed than prednisolone, resulting in a higher effective blood concentration of prednisolone.
化学的特性
White or almost white, hygroscopic, crystalline powder.
使用
antiinflammatory
プレドニゾロンリン酸エステルナトリウム 上流と下流の製品情報
原材料
準備製品