ChemicalBook >제품 카탈로그 >L371,257

L371,257

L371,257 구조식 이미지

카스 번호:: 162042-44-6

상품명:: L371,257

동의어(영문):: 257;L-371;L371,257;L371,257,L 371,257;1-[1-[4-(1-acetylpiperidin-4-yl)oxy-2-methoxybenzoyl]piperidin-4-yl]-4H-3,1-benzoxazin-2-one;1-[4-[(1-Acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]-4-(2-oxo-2H-3,1-benzoxazin-1(4H)-yl)piperidine;2H-3,1-Benzoxazin-2-one, 1-[1-[4-[(1-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]-4-piperidinyl]-1,4-dihydro-

CBNumber:: CB8850593

분자식:: C28H33N3O6

포뮬러 무게:: 507.58

MOL 파일:: 162042-44-6.mol

속성

안전

용도

공급 업체 31

L371,257 속성

끓는 점: 728.9±60.0 °C(Predicted)

밀도: 1.282±0.06 g/cm3(Predicted)

저장 조건: Store at RT

용해도: Soluble to 10 mM in DMSO with gentle warming

물리적 상태: 가루

산도 계수 (pKa): 0.73±0.20(Predicted)

안전

L371,257 C화학적 특성, 용도, 생산

용도

L-371,257 is a potent antagonist of oxytocin-induced contractions of the rat uterus in vitro and in vivo and has significant oral bioavailability in rats.

생물학적 활성

Potent, high affinity human oxytocin (OT) receptor antagonist (K i = 4.6 nM) that displays > 800-fold selectivity over human arginine vasopressin receptors V 1a and V 2 . Antagonizes oxytocin-induced contractions in isolated rat uterine tissue (pA 2 = 8.44) and in anesthetised rats following intravenous and intraduodenal administration. Orally active.

L371,257 준비 용품 및 원자재

원자재

준비 용품

L371,257 공급 업체

글로벌( 31)공급 업체

공급자	전화	이메일	국가	제품 수	이점
TargetMol Chemicals Inc.	+1-781-999-5354 +1-00000000000	marketing@targetmol.com	United States	19892	58
Nantong HI-FUTURE Biology Co., Ltd.	+undefined18051384581	sales@chemhifuture.com	China	3136	58
Wuhan Topule Biopharmaceutical Co., Ltd	+8618327326525	masar@topule.com	China	8474	58
Aladdin Scientific	+1-833-552-7181	sales@aladdinsci.com	United States	57511	58
3B Pharmachem (Wuhan) International Co.,Ltd.	821-50328103-801 18930552037	3bsc@sina.com	China	15848	69
EMMX Biotechnology LLC	888-539-0666	info@emmx.com	United States	8449	60
Beijing Solarbio Science & Tecnology Co., Ltd.	010-50973130 4009686088	3193328036@qq.com	China	29797	68
Hebei Weite Medical Technology Co., Ltd	13180081292	contact@wetogethermed.com	China	7273	58
Nantong Hi-Future Biotechnology Co., Ltd	18051384581	sales@chemhifuture.com	China	2996	58
Shanghai Universal Biotech Co.,Ltd	18768175414	gaojun@univ-bio.com	China	24998	58

L371,257 관련 검색:

4-Cbz-Aminopiperidine 1-Acetyl-4-(methylamino)piperidine 4-Methoxysalicylamide 4-(4-METHYLPHENOXY)PIPERIDINE HYDROCHLORIDE 4-PHENOXYPIPERIDINE 4-[3-(Dimethylamino)propoxy]benzaldehyde 1-(4-ISOPROPOXYPHENYL)METHANAMINE 2,4-Dihydroxybenzamide 4-ANILINO-1-BENZYLPIPERIDINE 4-(3-METHOXYPHENOXY)PIPERIDINE 1-Acetylpiperidin-4-amine 4-(PIPERIDIN-4-YLOXY)BENZAMIDE (4-AMINO-PIPERIDIN-1-YL)-PHENYL-METHANONE Benzamide, N-(3-dimethylaminopropyl)-p-propoxy- 4-ETHOXY-N,N-DIETHYLBENZAMIDE CHEMBRDG-BB 9072047 4-AMINOCARBETHOXYPIPERIDINE 1-ACETYLPIPERIDIN-4-OL