Cenicriviroc
|
- $60 - $20790
- Product name: Cenicriviroc
- CAS: 497223-25-3
- MF: C41H52N4O4S
- MW: 696.94
- EINECS:
- MDL Number:MFCD28502076
- Synonyms:Cenicriviroc;TAK652;Cenicriviroc mesylate (TAK-652);Cenicriviroc(TAK652);TAK-652; TAK652; TAK 652; TBR-652; TBR 652; TBR652; CENICRIVIROC.;CS-2572;TAK-652; TBR-652; TAK652; TBR652; TAK 652; TBR 652;TBR 652
43 prices
Selected condition：
Brand
- Abosyn
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Axon Medchem
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- TRC
Package
- 50mg
- 10mM*1mLinDMSO(Solid+Solvent)
- 1mg
- 250mg
- 10mM*1mLinDMSO(Solution)
- 10mM*1mLinDMSO
- 500μg
- 25mg
- 100mg
- 5MG
- 10mg
- 0.1g
- 0.25g
- 0.5g
- 1g
- 10g
- 1mL(10mMinDMSO)
- 5g
- ManufacturerAbosyn
- Product number90-2848
- Product description8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches)
- Packaging0.1g
- Price$314
- Updated2026-05-21
- Buy
- ManufacturerAbosyn
- Product number90-2848
- Product description8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches)
- Packaging0.25g
- Price$550
- Updated2026-05-21
- Buy
- ManufacturerAbosyn
- Product number90-2848
- Product description8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches)
- Packaging0.5g
- Price$943
- Updated2026-05-21
- Buy
- ManufacturerAbosyn
- Product number90-2848
- Product description8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches)
- Packaging1g
- Price$1078
- Updated2026-05-21
- Buy
- ManufacturerAbosyn
- Product number90-2848
- Product description8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches)
- Packaging5g
- Price$3234
- Updated2026-05-21
- Buy
- ManufacturerAbosyn
- Product number90-2848
- Product description8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches)
- Packaging10g
- Price$4528
- Updated2026-05-21
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberINB0005543
- Product descriptionCENICRIVIROC 95.00%
- Packaging5MG
- Price$500.98
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberBA1897
- Product descriptionCenicriviroc
- Packaging10mg
- Price$351
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA1897
- Product descriptionCenicriviroc
- Packaging1mL(10mMinDMSO)
- Price$386
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA1897
- Product descriptionCenicriviroc
- Packaging25mg
- Price$522
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA1897
- Product descriptionCenicriviroc
- Packaging50mg
- Price$711
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA1897
- Product descriptionCenicriviroc
- Packaging5mg
- Price$225
- Updated2026-05-06
- Buy
- ManufacturerApexBio Technology
- Product numberBA1897
- Product descriptionCenicriviroc
- Packaging1mg
- Price$81
- Updated2026-05-06
- Buy
- ManufacturerArctom
- Product numberHY-14882
- Product descriptionCenicriviroc 99.51%
- Packaging5mg
- Price$168
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-14882
- Product descriptionCenicriviroc 99.51%
- Packaging10mM*1mLinDMSO(Solid+Solvent)
- Price$245
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-14882
- Product descriptionCenicriviroc 99.51%
- Packaging10mM*1mLinDMSO(Solution)
- Price$257
- Updated2026-05-26
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| Abosyn | 90-2848 | 8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches) | 0.1g | $314 | 2026-05-21 | Buy |
| Abosyn | 90-2848 | 8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches) | 0.25g | $550 | 2026-05-21 | Buy |
| Abosyn | 90-2848 | 8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches) | 0.5g | $943 | 2026-05-21 | Buy |
| Abosyn | 90-2848 | 8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches) | 1g | $1078 | 2026-05-21 | Buy |
| Abosyn | 90-2848 | 8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches) | 5g | $3234 | 2026-05-21 | Buy |
| Abosyn | 90-2848 | 8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1,2,3,4-tetrahydrobenzo[b]azocine-5-carboxamide >95%(Puritymayvarybetweenbatches) | 10g | $4528 | 2026-05-21 | Buy |
| American Custom Chemicals Corporation | INB0005543 | CENICRIVIROC 95.00% | 5MG | $500.98 | 2021-12-16 | Buy |
| ApexBio Technology | BA1897 | Cenicriviroc | 10mg | $351 | 2026-05-06 | Buy |
| ApexBio Technology | BA1897 | Cenicriviroc | 1mL(10mMinDMSO) | $386 | 2026-05-06 | Buy |
| ApexBio Technology | BA1897 | Cenicriviroc | 25mg | $522 | 2026-05-06 | Buy |
| ApexBio Technology | BA1897 | Cenicriviroc | 50mg | $711 | 2026-05-06 | Buy |
| ApexBio Technology | BA1897 | Cenicriviroc | 5mg | $225 | 2026-05-06 | Buy |
| ApexBio Technology | BA1897 | Cenicriviroc | 1mg | $81 | 2026-05-06 | Buy |
| Arctom | HY-14882 | Cenicriviroc 99.51% | 5mg | $168 | 2026-05-26 | Buy |
| Arctom | HY-14882 | Cenicriviroc 99.51% | 10mM*1mLinDMSO(Solid+Solvent) | $245 | 2026-05-26 | Buy |
| Arctom | HY-14882 | Cenicriviroc 99.51% | 10mM*1mLinDMSO(Solution) | $257 | 2026-05-26 | Buy |
Properties
Boiling point :913.5±65.0 °C(Predicted)
Density :1.17±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMF: 20 mg/ml; DMSO: 20 mg/ml; DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml; Ethanol: 5 mg/ml
form :A crystalline solid
pka :12.96±0.70(Predicted)
color :Light yellow to yellow
Density :1.17±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMF: 20 mg/ml; DMSO: 20 mg/ml; DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml; Ethanol: 5 mg/ml
form :A crystalline solid
pka :12.96±0.70(Predicted)
color :Light yellow to yellow
Safety Information
| Symbol(GHS): |
|
|||||||||||||||||||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Signal word: | Warning | |||||||||||||||||||||||||||||||||||
| Hazard statements: |
|
|||||||||||||||||||||||||||||||||||
| Precautionary statements: |
|
Description
Cenicriviroc is a dual antagonist of chemokine receptor types 2 and 5 (CCR2/CCR5). The receptors are found on Kupffer cells and hepatic stellate cells, and preclinical studies suggest its anti-inflammatory and anti-fibrotic activity. In the phase 2b CENTAUR study, cenicriviroc treatment for 1 year failed to achieve the primary outcome of a decrease in NAFLD activity score by ≥2 points with no worsening of fibrosis. Nonetheless, one of the key secondary outcomes, improvement in liver fibrosis without worsening of NASH, was achieved in 20% in the treatment group, compared with 10% in the placebo group. Besides, cenicriviroc reduced the serum levels interleukin- 6, C-reactive protein and fibrinogen, suggesting its action on inflammation that may not be reflected by crude histological assessment. A phase 3 study is planned.Related product price
- Obeticholic Acid
$20-1872 - GDC-0068
$28-2964
