Cilastatin sodium
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- $39 - $2450
- Product name: Cilastatin sodium
- CAS: 81129-83-1
- MF: C16H25N2O5S.Na
- MW: 380.44
- EINECS:279-694-4
- MDL Number:MFCD08459332
- Synonyms:Cilastatine;Cilastatin sodium;Sodium 7-(2-amino-2-carboxy-ethyl)sulfanyl-2-(2,2-dimethylcyclopropyl)carbonylamino-hept-2-enoate;Sodium hydrogen 7-[(2-amino-2-carboxylatoethyl)thio]-2-[[(2,2-dimethylcyclopropyl)carbonyl]amino]hept-2-enoate;Sodium Cilastatin;[R-[R*,S*-(Z)]]-7-[(2-Amino-2-carboxyethyl)thio]-2-[[(2,2-dimethylcyclopropyl)carbonyl]amino]-2-heptenoic acid monosodium salt;(Z)-7-[(R)-2-Amino-2-carboxyethylthio]-2-[(S)-2,2-dimethylcyclopropylcarbonylamino]-2-heptenoic acid 1-sodium salt;(2Z)-7-[[(2R)-2-Amino-2-carboxyethyl]thio]-2-[[[(1S)-2,2-dimethylcyclopropyl]carbonyl]amino]-2-heptenoicacidsodiumsalt
26 prices
Selected condition：
Brand
- AHH
- AK Scientific
- American Custom Chemicals Corporation
- AvaChem
- Biosynth Carbosynth
- Chem-Impex
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TCI Chemical
- TRC
Package
- 25mg
- c2170000
- 10MG
- 50mg
- 100mg
- 250mg
- 500mg
- 1G
- 2ml
- 5g
- 10g
- 25 mg
- ManufacturerAHH
- Product numberMT-49258
- Product descriptionCilastatin sodium 99%
- Packaging5g
- Price$630
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product numberI422
- Product descriptionCilastatin sodium
- Packaging50mg
- Price$350
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0002011
- Product descriptionCILASTATIN SODIUM 95.00%
- Packaging10MG
- Price$641.55
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0002011
- Product descriptionCILASTATIN SODIUM 95.00%
- Packaging1G
- Price$825.3
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0002011
- Product descriptionCILASTATIN SODIUM 95.00%
- Packaging50MG
- Price$952.01
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number1721
- Product descriptionCilastatin sodium salt
- Packaging25mg
- Price$39
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number1721
- Product descriptionCilastatin sodium salt
- Packaging100mg
- Price$79
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number1721
- Product descriptionCilastatin sodium salt
- Packaging250mg
- Price$189
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number1721
- Product descriptionCilastatin sodium salt
- Packaging1g
- Price$349
- Updated2021-12-16
- Buy
- ManufacturerAvaChem
- Product number1721
- Product descriptionCilastatin sodium salt
- Packaging10g
- Price$2450
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBC164306
- Product descriptionCilastatin sodium
- Packaging10mg
- Price$65
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFC61442
- Product descriptionCilastatin sodium
- Packaging25mg
- Price$75
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFC61442
- Product descriptionCilastatin sodium
- Packaging50mg
- Price$100
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFC61442
- Product descriptionCilastatin sodium
- Packaging100mg
- Price$150
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFC61442
- Product descriptionCilastatin sodium
- Packaging250mg
- Price$250
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBC164306
- Product descriptionCilastatin sodium
- Packaging100mg
- Price$250
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AHH | MT-49258 | Cilastatin sodium 99% | 5g | $630 | 2021-12-16 | Buy |
| AK Scientific | I422 | Cilastatin sodium | 50mg | $350 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0002011 | CILASTATIN SODIUM 95.00% | 10MG | $641.55 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0002011 | CILASTATIN SODIUM 95.00% | 1G | $825.3 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0002011 | CILASTATIN SODIUM 95.00% | 50MG | $952.01 | 2021-12-16 | Buy |
| AvaChem | 1721 | Cilastatin sodium salt | 25mg | $39 | 2021-12-16 | Buy |
| AvaChem | 1721 | Cilastatin sodium salt | 100mg | $79 | 2021-12-16 | Buy |
| AvaChem | 1721 | Cilastatin sodium salt | 250mg | $189 | 2021-12-16 | Buy |
| AvaChem | 1721 | Cilastatin sodium salt | 1g | $349 | 2021-12-16 | Buy |
| AvaChem | 1721 | Cilastatin sodium salt | 10g | $2450 | 2021-12-16 | Buy |
| Biosynth Carbosynth | BC164306 | Cilastatin sodium | 10mg | $65 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FC61442 | Cilastatin sodium | 25mg | $75 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FC61442 | Cilastatin sodium | 50mg | $100 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FC61442 | Cilastatin sodium | 100mg | $150 | 2021-12-16 | Buy |
| Biosynth Carbosynth | FC61442 | Cilastatin sodium | 250mg | $250 | 2021-12-16 | Buy |
| Biosynth Carbosynth | BC164306 | Cilastatin sodium | 100mg | $250 | 2021-12-16 | Buy |
Properties
Melting point :>160°C (dec.)
Flash point :87℃
storage temp. :2-8°C
solubility :Very soluble in water and in methanol, slightly soluble in anhydrous ethanol, very slightly soluble in dimethyl sulfoxide, practically insoluble in acetone and in methylene chloride.
form :Solid
pka :pKa1 2.0; pKa2 4.4; pKa3 9.2(at 25℃)
color :White
biological source :synthetic (organic)
Water Solubility :water: 10mg/mL, clear, colorless to faintly yellow
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.
InChIKey :QXPBTTUOVWMPJN-LZTDVXLXNA-M
SMILES :[C@H]1(C(=O)N/C(=C\CCCCSC[C@H](N)C(O)=O)/C(=O)[O-])CC1(C)C.[Na+] |&1:0,12,r|
CAS DataBase Reference :81129-83-1(CAS DataBase Reference)
Flash point :87℃
storage temp. :2-8°C
solubility :Very soluble in water and in methanol, slightly soluble in anhydrous ethanol, very slightly soluble in dimethyl sulfoxide, practically insoluble in acetone and in methylene chloride.
form :Solid
pka :pKa1 2.0; pKa2 4.4; pKa3 9.2(at 25℃)
color :White
biological source :synthetic (organic)
Water Solubility :water: 10mg/mL, clear, colorless to faintly yellow
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO or ethanol may be stored at -20°C for up to 1 month.
InChIKey :QXPBTTUOVWMPJN-LZTDVXLXNA-M
SMILES :[C@H]1(C(=O)N/C(=C\CCCCSC[C@H](N)C(O)=O)/C(=O)[O-])CC1(C)C.[Na+] |&1:0,12,r|
CAS DataBase Reference :81129-83-1(CAS DataBase Reference)
Safety Information
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| Signal word: | Warning | ||||||||||||||
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Description
Cilastatin Na (81129-83-1) is a dehydropeptidase-1 inhibitor. Inhibits the proteolytic conversion of leukotriene D4to E4.1 Inhibits the mammalian β-lactamase renal dipeptidase (dehydropeptidase-1, DPEP1) and thus is used as an antibacterial adjunct to extend the half-life of β-lactam antibiotics.2Cilastatin also inhibits bacterial metallo-β-lactamase and thereby may block resistance to the carbapenem family of antibiotics in certain bacteria.3 Suppresses invasion and metastasis of DPEP1-expressing tumor cells.4More related product prices
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