Desmethyl loperamide
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- $203 - $3281.5
- Product name: Desmethyl loperamide
- CAS: 66164-07-6
- MF: C28H31ClN2O2
- MW: 463.01
- EINECS:
- MDL Number:MFCD08063667
- Synonyms:4-(4-Chlorophenyl)-4-hydroxy-N-methyl-a,a-diphenyl-1-piperidinebutanamide;N-Desmethyl Loperamide;R 20905;Desmethyl loperamide HCl;Desmethylloperamide D5;4-(4-Chlorophenyl)-4-hydroxy-N-Methyl-α,α-diphenyl-1-piperidinebutanaMide;1-Piperidinebutanamide, 4-(4-chlorophenyl)-4-hydroxy-N-methyl-α,α-diphenyl-;dLop
22 prices
Selected condition：
Brand
- aablocks
- AK Scientific
- American Custom Chemicals Corporation
- Biosynth
- Cayman Chemical
- ChemScene
- TRC
- Usbiological
Package
- 0.025mg
- 0.05mg
- 0.1mg
- 0.25mg
- 0.5mg
- 500μg
- 1mg
- 2mg
- 5mg
- 10MG
- 25mg
- 500??g
- Manufactureraablocks
- Product numberAA00F9ZC
- Product description4-(4-Chlorophenyl)-4-hydroxy-N-methyl-α,α-diphenyl-1-piperidinebutanamide ≥98%
- Packaging1mg
- Price$363
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00F9ZC
- Product description4-(4-Chlorophenyl)-4-hydroxy-N-methyl-α,α-diphenyl-1-piperidinebutanamide ≥98%
- Packaging5mg
- Price$1083
- Updated2026-05-28
- Buy
- ManufacturerAK Scientific
- Product number3134CR
- Product descriptionN-Desmethylloperamide
- Packaging5mg
- Price$1193
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006893
- Product descriptionDESMETHYL LOPERAMIDE 95.00%
- Packaging1MG
- Price$438.9
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0006893
- Product descriptionDESMETHYL LOPERAMIDE 95.00%
- Packaging10MG
- Price$2055.9
- Updated2021-12-16
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging25mg
- Price$3281.5
- Updated2021-12-16
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging2mg
- Price$528.6
- Updated2021-12-16
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging1mg
- Price$290.7
- Updated2021-12-16
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging10mg
- Price$1747.2
- Updated2021-12-16
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging0.025mg
- Price$900
- Updated2026-06-04
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging0.05mg
- Price$900
- Updated2026-06-04
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging0.1mg
- Price$900
- Updated2026-06-04
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging0.25mg
- Price$900
- Updated2026-06-04
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging0.5mg
- Price$900
- Updated2026-06-04
- Buy
- ManufacturerBiosynth
- Product numberFD21287
- Product descriptionN-Desmethyl loperamide
- Packaging5mg
- Price$961
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number16126
- Product descriptionN-desmethyl Loperamide ≥98%
- Packaging5mg
- Price$1083
- Updated2026-04-30
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA00F9ZC | 4-(4-Chlorophenyl)-4-hydroxy-N-methyl-α,α-diphenyl-1-piperidinebutanamide ≥98% | 1mg | $363 | 2026-05-28 | Buy |
| aablocks | AA00F9ZC | 4-(4-Chlorophenyl)-4-hydroxy-N-methyl-α,α-diphenyl-1-piperidinebutanamide ≥98% | 5mg | $1083 | 2026-05-28 | Buy |
| AK Scientific | 3134CR | N-Desmethylloperamide | 5mg | $1193 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0006893 | DESMETHYL LOPERAMIDE 95.00% | 1MG | $438.9 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0006893 | DESMETHYL LOPERAMIDE 95.00% | 10MG | $2055.9 | 2021-12-16 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 25mg | $3281.5 | 2021-12-16 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 2mg | $528.6 | 2021-12-16 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 1mg | $290.7 | 2021-12-16 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 10mg | $1747.2 | 2021-12-16 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 0.025mg | $900 | 2026-06-04 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 0.05mg | $900 | 2026-06-04 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 0.1mg | $900 | 2026-06-04 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 0.25mg | $900 | 2026-06-04 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 0.5mg | $900 | 2026-06-04 | Buy |
| Biosynth | FD21287 | N-Desmethyl loperamide | 5mg | $961 | 2021-12-16 | Buy |
| Cayman Chemical | 16126 | N-desmethyl Loperamide ≥98% | 5mg | $1083 | 2026-04-30 | Buy |
Properties
Melting point :219-221C
Boiling point :678.3±55.0 °C(Predicted)
Density :1+-.0.06 g/cm3(Predicted)
storage temp. :-20°C Freezer
solubility :DMF: 2 mg/ml; DMF:PBS(pH 7.2)(1:1): 0.5 mg/ml; DMSO: 1 mg/ml
form :A crystalline solid
pka :13.85±0.20(Predicted)
Boiling point :678.3±55.0 °C(Predicted)
Density :1+-.0.06 g/cm3(Predicted)
storage temp. :-20°C Freezer
solubility :DMF: 2 mg/ml; DMF:PBS(pH 7.2)(1:1): 0.5 mg/ml; DMSO: 1 mg/ml
form :A crystalline solid
pka :13.85±0.20(Predicted)
Safety Information
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| Signal word: | Danger | ||||||||||||||||
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Description
Loperamide is an opiate which potently and selectively activates μ opioid receptors (Ki = 0.16 nM) exclusively in the periphery. N-Desmethyl-loperamide (dLop) is a major metabolite of loperamide. Like loperamide, dLop is a substrate of the ATP-dependent efflux transporter, P-glycoprotein. As a result, both the parent compound and the metabolite display restricted passage through the blood-brain barrier. dLop in biological samples can be analyzed by a variety of methods.Related product price
Suppliers and manufacturers
J & K SCIENTIFIC LTD.
Chemsky（shanghai）International Co.,Ltd.
Daicel Chiral Technologies (China)CO.,LTD
Artis Chemistry (Shanghai) Co. Ltd.
Finetech Industry Limited
BOC Sciences
Shanghai Chaolan Chemical Technology Center
Amadis Chemical Company Limited
Shenzhen Polymeri Biochemical Technology Co., Ltd.
Hefei Molake Biotechnology Co., Ltd.