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ChemicalBook CAS DataBase List methyl (2E)-3-[6-(trifluoromethyl)pyridin-3-yl]prop-2-enoate
1119807-17-8

methyl (2E)-3-[6-(trifluoromethyl)pyridin-3-yl]prop-2-enoate synthesis

3synthesis methods
21204-67-1 Synthesis
methyl (triphenylphosphoranylidene)acetate

21204-67-1
23 suppliers
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386704-12-7 Synthesis
6-(TRIFLUOROMETHYL)PYRIDINE-3-CARBOXALDEHYDE

386704-12-7
195 suppliers
$6.00/100mg

methyl (2E)-3-[6-(trifluoromethyl)pyridin-3-yl]prop-2-enoate

1119807-17-8
5 suppliers
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-

Yield:1119807-17-8 99%

Reaction Conditions:

in dichloromethane at 0 - 20; for 4 h;Wittig Olefination;

References:

Meyers, Marvin J.;Liu, Jianguang;Xu, Jing;Leng, Fang;Guan, Jiantong;Liu, Zhijun;McNitt, Sarah A.;Qin, Limei;Dai, Linglin;Ma, Hongwei;Adah, Dickson;Zhao, Siting;Li, Xiaofen;Polino, Alex J.;Nasamu, Armiyaw S.;Goldberg, Daniel E.;Liu, Xiaorong;Lu, Yongzhi;Tu, Zhengchao;Chen, Xiaoping;Tortorella, Micky D. [Journal of Medicinal Chemistry,2019,vol. 62,# 7,p. 3503 - 3512] Location in patent:supporting information

5927-18-4 Synthesis
Trimethyl phosphonoacetate

5927-18-4
331 suppliers
$5.00/25g

386704-12-7 Synthesis
6-(TRIFLUOROMETHYL)PYRIDINE-3-CARBOXALDEHYDE

386704-12-7
195 suppliers
$6.00/100mg

methyl (2E)-3-[6-(trifluoromethyl)pyridin-3-yl]prop-2-enoate

1119807-17-8
5 suppliers
inquiry

acrylic acid methyl ester

292638-85-8
5 suppliers
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436799-32-5 Synthesis
2-Trifluoromethyl-5-bromopyridine

436799-32-5
325 suppliers
$5.00/250mg

methyl (2E)-3-[6-(trifluoromethyl)pyridin-3-yl]prop-2-enoate

1119807-17-8
5 suppliers
inquiry