α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyridinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-benzeneacetonitrile
![α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyridinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-benzeneacetonitrile price.](/CAS/20211123/GIF/853910-02-8.gif)
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- $37 - $3580.2
- Product name: α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyridinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-benzeneacetonitrile
- CAS: 853910-02-8
- MF: C28H21N5
- MW: 427.51
- EINECS:200-258-5
- MDL Number:MFCD16618394
- Synonyms:BAG 956;α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyridinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-benzeneacetonitrile;2-Methyl-2-[4-[2-methyl-8-[(pyridin-3-yl)ethynyl]imidazo[4,5-c]quinolin-1-yl]phenyl]propionitrile;2-Methyl-2-[4-(2-methyl-8-pyridin-3-ylethynyl-imidazo[4,5-c]quinolin-1-yl)-phenyl]-propionitrile,NVP-BAG;NVP-BAG 956 BAG 956;NVP-BAG956, >=98%;BAG956(NVP-BAG956);NVP-BAG956;BAG 956;NVP-BAG 956
23 prices
Selected condition：
Brand
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Axon Medchem
- Biorbyt Ltd
- Cayman Chemical
- Crysdot
- DC Chemicals
- Medical Isotopes, Inc.
- Sigma-Aldrich
- Tocris
- TRC
- Usbiological
Package
- 50
- 10
- 1mg
- 5mg
- 10MG
- 2x5mg
- 50MG
- 100mg
- 250mg
- 1g
- 1000mg
- ManufacturerAK Scientific
- Product numberX5814
- Product description2-Methyl-2-{4-[2-methyl-8-(pyridin-3-ylethynyl)-1H-imidazo[4,5-c]quinolin-1-yl]phenyl}propanenitrile
- Packaging5mg
- Price$266
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0013704
- Product descriptionA,A-DIMETHYL-4-[2-METHYL-8-[2-(3-PYRIDINYL)ETHYNYL]-1H-IMIDAZO[4,5-C]QUINOLIN-1-YL]-BENZENEACETONITRILE 95.00%
- Packaging5MG
- Price$257.4
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0013704
- Product descriptionA,A-DIMETHYL-4-[2-METHYL-8-[2-(3-PYRIDINYL)ETHYNYL]-1H-IMIDAZO[4,5-C]QUINOLIN-1-YL]-BENZENEACETONITRILE 95.00%
- Packaging10MG
- Price$807.35
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0013704
- Product descriptionA,A-DIMETHYL-4-[2-METHYL-8-[2-(3-PYRIDINYL)ETHYNYL]-1H-IMIDAZO[4,5-C]QUINOLIN-1-YL]-BENZENEACETONITRILE 95.00%
- Packaging50MG
- Price$1558.1
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA3672
- Product descriptionNVP-BAG956
- Packaging5mg
- Price$386
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA3672
- Product descriptionNVP-BAG956
- Packaging10mg
- Price$693
- Updated2021-12-16
- Buy
- ManufacturerAxon Medchem
- Product numberAxon1282
- Product descriptionBAG956-NVP-BAG956 99%
- Packaging2x5mg
- Price$154
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181101
- Product descriptionNVP-BAG956(BAG 956) >98%
- Packaging100mg
- Price$912.9
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181101
- Product descriptionNVP-BAG956(BAG 956) >98%
- Packaging250mg
- Price$1802
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb181101
- Product descriptionNVP-BAG956(BAG 956) >98%
- Packaging1000mg
- Price$3580.2
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number24195
- Product descriptionNVP-BAG956 ≥98%
- Packaging1mg
- Price$37
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number24195
- Product descriptionNVP-BAG956 ≥98%
- Packaging5mg
- Price$151
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number24195
- Product descriptionNVP-BAG956 ≥98%
- Packaging10mg
- Price$231
- Updated2024-03-01
- Buy
- ManufacturerCrysdot
- Product numberCD31000594
- Product descriptionNVP-BAG956(BAG956) 98+%
- Packaging10mg
- Price$107
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD31000594
- Product descriptionNVP-BAG956(BAG956) 98+%
- Packaging50mg
- Price$487
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC7250
- Product descriptionNVP-BAG956(BAG956) >98%
- Packaging250mg
- Price$1200
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | X5814 | 2-Methyl-2-{4-[2-methyl-8-(pyridin-3-ylethynyl)-1H-imidazo[4,5-c]quinolin-1-yl]phenyl}propanenitrile | 5mg | $266 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0013704 | A,A-DIMETHYL-4-[2-METHYL-8-[2-(3-PYRIDINYL)ETHYNYL]-1H-IMIDAZO[4,5-C]QUINOLIN-1-YL]-BENZENEACETONITRILE 95.00% | 5MG | $257.4 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0013704 | A,A-DIMETHYL-4-[2-METHYL-8-[2-(3-PYRIDINYL)ETHYNYL]-1H-IMIDAZO[4,5-C]QUINOLIN-1-YL]-BENZENEACETONITRILE 95.00% | 10MG | $807.35 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0013704 | A,A-DIMETHYL-4-[2-METHYL-8-[2-(3-PYRIDINYL)ETHYNYL]-1H-IMIDAZO[4,5-C]QUINOLIN-1-YL]-BENZENEACETONITRILE 95.00% | 50MG | $1558.1 | 2021-12-16 | Buy |
| ApexBio Technology | A3672 | NVP-BAG956 | 5mg | $386 | 2021-12-16 | Buy |
| ApexBio Technology | A3672 | NVP-BAG956 | 10mg | $693 | 2021-12-16 | Buy |
| Axon Medchem | Axon1282 | BAG956-NVP-BAG956 99% | 2x5mg | $154 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181101 | NVP-BAG956(BAG 956) >98% | 100mg | $912.9 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181101 | NVP-BAG956(BAG 956) >98% | 250mg | $1802 | 2021-12-16 | Buy |
| Biorbyt Ltd | orb181101 | NVP-BAG956(BAG 956) >98% | 1000mg | $3580.2 | 2021-12-16 | Buy |
| Cayman Chemical | 24195 | NVP-BAG956 ≥98% | 1mg | $37 | 2024-03-01 | Buy |
| Cayman Chemical | 24195 | NVP-BAG956 ≥98% | 5mg | $151 | 2024-03-01 | Buy |
| Cayman Chemical | 24195 | NVP-BAG956 ≥98% | 10mg | $231 | 2024-03-01 | Buy |
| Crysdot | CD31000594 | NVP-BAG956(BAG956) 98+% | 10mg | $107 | 2021-12-16 | Buy |
| Crysdot | CD31000594 | NVP-BAG956(BAG956) 98+% | 50mg | $487 | 2021-12-16 | Buy |
| DC Chemicals | DC7250 | NVP-BAG956(BAG956) >98% | 250mg | $1200 | 2021-12-16 | Buy |
Properties
Melting point :>224oC (dec.)
Boiling point :694.8±65.0 °C(Predicted)
Density :1.17
storage temp. :Store at RT
solubility :DMSO (Slightly, Heated), Methanol (Slightly)
form :Orange powder
pka :4.99±0.30(Predicted)
color :White
Boiling point :694.8±65.0 °C(Predicted)
Density :1.17
storage temp. :Store at RT
solubility :DMSO (Slightly, Heated), Methanol (Slightly)
form :Orange powder
pka :4.99±0.30(Predicted)
color :White
Safety Information
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Description
BAG 956 is a dual PDK1 and class I PI 3-kinase inhibitor (IC50 values are 245, 56, 446, 35 and 117 nM for PDK1 and PI3K p110 -α, -β, -δ, and -γ respectively). BAG 956 has been shown to inhibit cellular AKT phosphorylation at Thr308. BAG 956 also blocks cell proliferation and causes arrest in the G1 phase of the cell cycle. BAG 956 has been shown to slow tumor progression in mouse xenograft models.Suppliers and manufacturers
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J & K SCIENTIFIC LTD.
3B Pharmachem (Wuhan) International Co.,Ltd.
Chembest Research Laboratories Limited
