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ChemicalBook >> CAS DataBase List >> Relugolix

Relugolix

Relugolix price.
  • $16 - $3728.1
  • Product name: Relugolix
  • CAS: 737789-87-6
  • MF: C29H27F2N7O5S
  • MW: 623.63
  • EINECS:237-099-7
  • MDL Number:MFCD25976856
  • Synonyms:TKA-385 Relugolix;TAK-385,Relugolix;CS-2851;TAK-385;TAK 385;TAK385;1-[4-[1-[(2,6-difluorophenyl)methyl]-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-3-methoxyurea;10G,100G,500G,1KG;N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxy urea;1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydro thieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxy urea, Relugolix
69 prices
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  • aablocks
  • ACHEMBLOCK
  • AK Scientific
  • Ambeed
  • Arctom
  • Biorbyt Ltd
  • Cayman Chemical
  • ChemScene
  • Crysdot
  • DC Chemicals
  • Matrix Scientific
Package
  • 5mg
  • 10mM*1mLinDMSO(Solution)
  • 1mg
  • 10mM*1mLinDMSO(Solid+Solvent)
  • 10mg
  • 25mg
  • 25.00mg
  • 50.00mg
  • 50mg
  • 100mg
  • 100.00mg
  • 250mg
  • 1g
  • 5g
  • 10g
  • Manufactureraablocks
  • Product numberAA00FBYA
  • Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
  • Packaging25mg
  • Price$50
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00FBYA
  • Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
  • Packaging50mg
  • Price$84
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00FBYA
  • Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea ≥98%
  • Packaging5mg
  • Price$16
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00FBYA
  • Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
  • Packaging100mg
  • Price$128
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00FBYA
  • Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
  • Packaging250mg
  • Price$230
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00FBYA
  • Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
  • Packaging1g
  • Price$458
  • Updated2026-05-28
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  • Manufactureraablocks
  • Product numberAA00FBYA
  • Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
  • Packaging5g
  • Price$1580
  • Updated2026-05-28
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  • ManufacturerACHEMBLOCK
  • Product numberQ65610
  • Product description1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea 98%
  • Packaging25MG
  • Price$215
  • Updated2026-05-27
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  • ManufacturerACHEMBLOCK
  • Product numberQ65610
  • Product description1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea 98%
  • Packaging100MG
  • Price$540
  • Updated2026-05-27
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  • ManufacturerAK Scientific
  • Product number6863CR
  • Product descriptionRelugolix
  • Packaging25mg
  • Price$691
  • Updated2021-12-16
  • Buy
  • ManufacturerAK Scientific
  • Product number6863CR
  • Product descriptionRelugolix
  • Packaging10mg
  • Price$370
  • Updated2021-12-16
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  • ManufacturerAmbeed
  • Product numberA261708
  • Product descriptionRelugolix 98%
  • Packaging250mg
  • Price$290
  • Updated2026-06-05
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  • ManufacturerAmbeed
  • Product numberA261708
  • Product descriptionRelugolix 98%
  • Packaging100mg
  • Price$162
  • Updated2026-06-05
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  • ManufacturerAmbeed
  • Product numberA261708
  • Product descriptionRelugolix 98%
  • Packaging50mg
  • Price$106
  • Updated2026-06-05
  • Buy
  • ManufacturerAmbeed
  • Product numberA261708
  • Product descriptionRelugolix 98%
  • Packaging25mg
  • Price$63
  • Updated2026-06-05
  • Buy
  • ManufacturerAmbeed
  • Product numberA261708
  • Product descriptionRelugolix 98%
  • Packaging1g
  • Price$579
  • Updated2026-06-05
  • Buy
Manufacturer Product number Product description Packaging Price Updated Buy
aablocks AA00FBYA N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% 25mg $50 2026-05-28 Buy
aablocks AA00FBYA N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% 50mg $84 2026-05-28 Buy
aablocks AA00FBYA N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea ≥98% 5mg $16 2026-05-28 Buy
aablocks AA00FBYA N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% 100mg $128 2026-05-28 Buy
aablocks AA00FBYA N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% 250mg $230 2026-05-28 Buy
aablocks AA00FBYA N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% 1g $458 2026-05-28 Buy
aablocks AA00FBYA N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% 5g $1580 2026-05-28 Buy
ACHEMBLOCK Q65610 1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea 98% 25MG $215 2026-05-27 Buy
ACHEMBLOCK Q65610 1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea 98% 100MG $540 2026-05-27 Buy
AK Scientific 6863CR Relugolix 25mg $691 2021-12-16 Buy
AK Scientific 6863CR Relugolix 10mg $370 2021-12-16 Buy
Ambeed A261708 Relugolix 98% 250mg $290 2026-06-05 Buy
Ambeed A261708 Relugolix 98% 100mg $162 2026-06-05 Buy
Ambeed A261708 Relugolix 98% 50mg $106 2026-06-05 Buy
Ambeed A261708 Relugolix 98% 25mg $63 2026-06-05 Buy
Ambeed A261708 Relugolix 98% 1g $579 2026-06-05 Buy

Properties

Melting point :228 °C (decomp)(Solv: ethyl acetate (141-78-6); tetrahydrofuran (109-99-9))
Density :1.442±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO:20.0(Max Conc. mg/mL);32.1(Max Conc. mM)
Ethanol:1.0(Max Conc. mg/mL);1.6(Max Conc. mM) form :A crystalline solid
pka :13.17±0.70(Predicted)
color :White to off-white
InChIKey :AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES :N(C1=CC=C(C2SC3=C(C=2CN(C)C)C(=O)N(C2=NN=C(OC)C=C2)C(=O)N3CC2=C(F)C=CC=C2F)C=C1)C(NOC)=O

Safety Information

Symbol(GHS): Health Hazard (GHS08)
Signal word: Warning
Hazard statements:
Code Hazard statements Hazard class Category Signal word Pictogram P-Codes
H361 Suspected of damaging fertility or the unborn child Reproductive toxicity Category 2 Warning P201, P202, P281, P308+P313, P405,P501
H371 May cause damage to organs Specific target organ toxicity, single exposure Category 2 Warning P260, P264, P270, P309+P311, P405,P501
Precautionary statements:
P201 Obtain special instructions before use.
P202 Do not handle until all safety precautions have been read and understood.
P260 Do not breathe dust/fume/gas/mist/vapours/spray.
P264 Wash hands thoroughly after handling.
P264 Wash skin thouroughly after handling.
P270 Do not eat, drink or smoke when using this product.
P281 Use personal protective equipment as required.
P308+P313 IF exposed or concerned: Get medical advice/attention.
P309+P311 IF exposed or if you feel unwell: call a POISON CENTER or doctor/physician.
P405 Store locked up.
P501 Dispose of contents/container to..…

Description

Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. It possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al.

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