Relugolix
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- $32 - $3728.1
- Product name: Relugolix
- CAS: 737789-87-6
- MF: C29H27F2N7O5S
- MW: 623.63
- EINECS:237-099-7
- MDL Number:MFCD25976856
- Synonyms:TAK-385;TKA-385 Relugolix;TAK-385,Relugolix;CS-2851;TAK-385;TAK 385;TAK385;1-[4-[1-[(2,6-difluorophenyl)methyl]-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-3-methoxyurea;10G,100G,500G,1KG;N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxy urea
48 prices
Selected condition：
Brand
- AK Scientific
- Arctom
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- Matrix Scientific
Package
- 1mg
- 25.00mg
- 50.00mg
- 100.00mg
- 250mg
- 1g
- 10mM*1mLinDMSO(Solution)
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 10mM*1mLinDMSO(Solid+Solvent)
- ManufacturerAK Scientific
- Product number6863CR
- Product descriptionRelugolix
- Packaging10mg
- Price$370
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number6863CR
- Product descriptionRelugolix
- Packaging25mg
- Price$691
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberHY-16474R
- Product descriptionRelugolix (Standard)
- Packaging50mg
- Price$852
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474
- Product descriptionRelugolix 99.95%
- Packaging50mg
- Price$323
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberSLK-S5808
- Product descriptionRelugolix 99.76%
- Packaging25mg
- Price$447
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474
- Product descriptionRelugolix 99.95%
- Packaging100mg
- Price$523
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474R
- Product descriptionRelugolix (Standard)
- Packaging25mg
- Price$532
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474R
- Product descriptionRelugolix (Standard)
- Packaging10mg
- Price$266
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474
- Product descriptionRelugolix 99.95%
- Packaging5mg
- Price$67
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474
- Product descriptionRelugolix 99.95%
- Packaging10mM*1mLinDMSO(Solid+Solvent)
- Price$87
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474
- Product descriptionRelugolix 99.95%
- Packaging10mM*1mLinDMSO(Solution)
- Price$92
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474
- Product descriptionRelugolix 99.95%
- Packaging10mg
- Price$105
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberSLK-S5808
- Product descriptionRelugolix 99.76%
- Packaging5mg
- Price$140
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474R
- Product descriptionRelugolix (Standard)
- Packaging5mg
- Price$167
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474
- Product descriptionRelugolix 99.95%
- Packaging25mg
- Price$209
- Updated2026-05-26
- Buy
- ManufacturerArctom
- Product numberHY-16474R
- Product descriptionRelugolix (Standard)
- Packaging100mg
- Price$1277
- Updated2026-05-26
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 6863CR | Relugolix | 10mg | $370 | 2021-12-16 | Buy |
| AK Scientific | 6863CR | Relugolix | 25mg | $691 | 2021-12-16 | Buy |
| Arctom | HY-16474R | Relugolix (Standard) | 50mg | $852 | 2026-05-26 | Buy |
| Arctom | HY-16474 | Relugolix 99.95% | 50mg | $323 | 2026-05-26 | Buy |
| Arctom | SLK-S5808 | Relugolix 99.76% | 25mg | $447 | 2026-05-26 | Buy |
| Arctom | HY-16474 | Relugolix 99.95% | 100mg | $523 | 2026-05-26 | Buy |
| Arctom | HY-16474R | Relugolix (Standard) | 25mg | $532 | 2026-05-26 | Buy |
| Arctom | HY-16474R | Relugolix (Standard) | 10mg | $266 | 2026-05-26 | Buy |
| Arctom | HY-16474 | Relugolix 99.95% | 5mg | $67 | 2026-05-26 | Buy |
| Arctom | HY-16474 | Relugolix 99.95% | 10mM*1mLinDMSO(Solid+Solvent) | $87 | 2026-05-26 | Buy |
| Arctom | HY-16474 | Relugolix 99.95% | 10mM*1mLinDMSO(Solution) | $92 | 2026-05-26 | Buy |
| Arctom | HY-16474 | Relugolix 99.95% | 10mg | $105 | 2026-05-26 | Buy |
| Arctom | SLK-S5808 | Relugolix 99.76% | 5mg | $140 | 2026-05-26 | Buy |
| Arctom | HY-16474R | Relugolix (Standard) | 5mg | $167 | 2026-05-26 | Buy |
| Arctom | HY-16474 | Relugolix 99.95% | 25mg | $209 | 2026-05-26 | Buy |
| Arctom | HY-16474R | Relugolix (Standard) | 100mg | $1277 | 2026-05-26 | Buy |
Properties
Melting point :228 °C (decomp)(Solv: ethyl acetate (141-78-6); tetrahydrofuran (109-99-9))
Density :1.442±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO:20.0(Max Conc. mg/mL);32.1(Max Conc. mM)
Ethanol:1.0(Max Conc. mg/mL);1.6(Max Conc. mM) form :A crystalline solid
pka :13.17±0.70(Predicted)
color :White to off-white
InChIKey :AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES :N(C1=CC=C(C2SC3=C(C=2CN(C)C)C(=O)N(C2=NN=C(OC)C=C2)C(=O)N3CC2=C(F)C=CC=C2F)C=C1)C(NOC)=O
Density :1.442±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO:20.0(Max Conc. mg/mL);32.1(Max Conc. mM)
Ethanol:1.0(Max Conc. mg/mL);1.6(Max Conc. mM) form :A crystalline solid
pka :13.17±0.70(Predicted)
color :White to off-white
InChIKey :AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES :N(C1=CC=C(C2SC3=C(C=2CN(C)C)C(=O)N(C2=NN=C(OC)C=C2)C(=O)N3CC2=C(F)C=CC=C2F)C=C1)C(NOC)=O
Safety Information
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| Signal word: | Warning | ||||||||||||||||||||||
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Description
Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. It possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al.More related product prices
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