Relugolix
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- $16 - $3728.1
- Product name: Relugolix
- CAS: 737789-87-6
- MF: C29H27F2N7O5S
- MW: 623.63
- EINECS:237-099-7
- MDL Number:MFCD25976856
- Synonyms:TKA-385 Relugolix;TAK-385,Relugolix;CS-2851;TAK-385;TAK 385;TAK385;1-[4-[1-[(2,6-difluorophenyl)methyl]-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-3-methoxyurea;10G,100G,500G,1KG;N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxy urea;1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydro thieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxy urea, Relugolix
55 prices
Selected condition:
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- Ambeed
- Arctom
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- Matrix Scientific
Package
- 5mg
- 10mM*1mLinDMSO(Solution)
- 1mg
- 10mM*1mLinDMSO(Solid+Solvent)
- 10mg
- 25mg
- 25.00mg
- 50mg
- 50.00mg
- 100mg
- 100.00mg
- 250mg
- 1g
- 5g
- 10g
- Manufactureraablocks
- Product numberAA00FBYA
- Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
- Packaging25mg
- Price$50
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00FBYA
- Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
- Packaging50mg
- Price$84
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00FBYA
- Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea ≥98%
- Packaging5mg
- Price$16
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00FBYA
- Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
- Packaging100mg
- Price$128
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00FBYA
- Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
- Packaging250mg
- Price$230
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00FBYA
- Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
- Packaging1g
- Price$458
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA00FBYA
- Product descriptionN-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98%
- Packaging5g
- Price$1580
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberQ65610
- Product description1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea 98%
- Packaging100MG
- Price$540
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberQ65610
- Product description1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea 98%
- Packaging25MG
- Price$215
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product number6863CR
- Product descriptionRelugolix
- Packaging10mg
- Price$370
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number6863CR
- Product descriptionRelugolix
- Packaging25mg
- Price$691
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA261708
- Product descriptionRelugolix 98%
- Packaging1g
- Price$579
- Updated2026-06-05
- Buy
- ManufacturerAmbeed
- Product numberA261708
- Product descriptionRelugolix 98%
- Packaging5g
- Price$1639
- Updated2026-06-05
- Buy
- ManufacturerAmbeed
- Product numberA261708
- Product descriptionRelugolix 98%
- Packaging10g
- Price$2623
- Updated2026-06-05
- Buy
- ManufacturerAmbeed
- Product numberA261708
- Product descriptionRelugolix 98%
- Packaging25mg
- Price$63
- Updated2026-06-05
- Buy
- ManufacturerAmbeed
- Product numberA261708
- Product descriptionRelugolix 98%
- Packaging250mg
- Price$290
- Updated2026-06-05
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA00FBYA | N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% | 25mg | $50 | 2026-05-28 | Buy |
| aablocks | AA00FBYA | N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% | 50mg | $84 | 2026-05-28 | Buy |
| aablocks | AA00FBYA | N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea ≥98% | 5mg | $16 | 2026-05-28 | Buy |
| aablocks | AA00FBYA | N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% | 100mg | $128 | 2026-05-28 | Buy |
| aablocks | AA00FBYA | N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% | 250mg | $230 | 2026-05-28 | Buy |
| aablocks | AA00FBYA | N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% | 1g | $458 | 2026-05-28 | Buy |
| aablocks | AA00FBYA | N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxyurea 98% | 5g | $1580 | 2026-05-28 | Buy |
| ACHEMBLOCK | Q65610 | 1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea 98% | 100MG | $540 | 2026-05-27 | Buy |
| ACHEMBLOCK | Q65610 | 1-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea 98% | 25MG | $215 | 2026-05-27 | Buy |
| AK Scientific | 6863CR | Relugolix | 10mg | $370 | 2021-12-16 | Buy |
| AK Scientific | 6863CR | Relugolix | 25mg | $691 | 2021-12-16 | Buy |
| Ambeed | A261708 | Relugolix 98% | 1g | $579 | 2026-06-05 | Buy |
| Ambeed | A261708 | Relugolix 98% | 5g | $1639 | 2026-06-05 | Buy |
| Ambeed | A261708 | Relugolix 98% | 10g | $2623 | 2026-06-05 | Buy |
| Ambeed | A261708 | Relugolix 98% | 25mg | $63 | 2026-06-05 | Buy |
| Ambeed | A261708 | Relugolix 98% | 250mg | $290 | 2026-06-05 | Buy |
Properties
Melting point :228 °C (decomp)(Solv: ethyl acetate (141-78-6); tetrahydrofuran (109-99-9))
Density :1.442±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO:20.0(Max Conc. mg/mL);32.1(Max Conc. mM)
Ethanol:1.0(Max Conc. mg/mL);1.6(Max Conc. mM) form :A crystalline solid
pka :13.17±0.70(Predicted)
color :White to off-white
InChIKey :AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES :N(C1=CC=C(C2SC3=C(C=2CN(C)C)C(=O)N(C2=NN=C(OC)C=C2)C(=O)N3CC2=C(F)C=CC=C2F)C=C1)C(NOC)=O
Density :1.442±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO:20.0(Max Conc. mg/mL);32.1(Max Conc. mM)
Ethanol:1.0(Max Conc. mg/mL);1.6(Max Conc. mM) form :A crystalline solid
pka :13.17±0.70(Predicted)
color :White to off-white
InChIKey :AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES :N(C1=CC=C(C2SC3=C(C=2CN(C)C)C(=O)N(C2=NN=C(OC)C=C2)C(=O)N3CC2=C(F)C=CC=C2F)C=C1)C(NOC)=O
Safety Information
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| Signal word: | Warning | ||||||||||||||||||||||
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Description
Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. It possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al.More related product prices
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