MLN9708
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- $9 - $10065.83
- Product name: MLN9708
- CAS: 1201902-80-8
- MF: C20H23BCl2N2O9
- MW: 517.12
- EINECS:-0
- MDL Number:MFCD18251437
- Synonyms:4-(carboxymethyl)-2-((R)-1-(2-(2,5-dichlorobenzamido)acetamido)-3-methylbutyl)-6-oxo-1,3,2-dioxaborinane-4-carboxylic acid;MLN9708;MLN9708,MLN-9708,MLN 9708;4-Carboxy-2-[(1R)-1-[[2-[(2,5-dichlorobenzoyl)amino]acetyl]amino]-3-methylbutyl]-6-oxo-1,3,2-dioxaborinane-4-acetic acid;4-Carboxy-2-[(1R)-1-[[2-[(2,5-dichlorobenzoyl)amino]acetyl]amino]-3-methylbutyl]-6-oxo-1,3,2-dioxaborinane-4-acetic acid MLN9708;MLN9708;MLN-9708;4-(Carboxymethyl)-2-((R)-1-(2-(2,5-dichlorobenzamido)acetamido)-3-methylbutyl)-6-oxo-1,3,2-dio;MLN 9708 analog
59 prices
Selected condition:
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Ark Pharm
- Axon Medchem
- Biosynth
- Cayman Chemical
- Crysdot
- Matrix Scientific
- TRC
Package
- 2mg
- 2x5mg
- 1unit
- EvaluationSample
- 20mg
- 25.00g
- 50.00g
- 100.00g
- 25 mg
- 10mM(in1mLDMSO)
- 1mg
- 5mg
- 10mg
- 25mg
- 50mg
- 100MG
- 250mg
- 500mg
- 1g
- Manufactureraablocks
- Product numberAA000QH1
- Product description4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99%
- Packaging1mg
- Price$9
- Updated2026-05-25
- Buy
- Manufactureraablocks
- Product numberAA000QH1
- Product description4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99%
- Packaging5mg
- Price$20
- Updated2026-05-25
- Buy
- Manufactureraablocks
- Product numberAA000QH1
- Product description4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99%
- Packaging10mg
- Price$32
- Updated2026-05-25
- Buy
- Manufactureraablocks
- Product numberAA000QH1
- Product description4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99%
- Packaging25mg
- Price$46
- Updated2026-05-25
- Buy
- Manufactureraablocks
- Product numberAA000QH1
- Product description4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99%
- Packaging50mg
- Price$55
- Updated2026-05-25
- Buy
- Manufactureraablocks
- Product numberAA000QH1
- Product description4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 95%
- Packaging250mg
- Price$258
- Updated2026-05-25
- Buy
- Manufactureraablocks
- Product numberAA000QH1
- Product description4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid ≥98%
- Packaging500mg
- Price$435
- Updated2026-05-25
- Buy
- Manufactureraablocks
- Product numberAA000QH1
- Product description4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid ≥98%
- Packaging1g
- Price$783
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberF-4808
- Product descriptionMLN9708 98%
- Packaging1G
- Price$495
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberF-4808
- Product descriptionMLN9708 98%
- Packaging25MG
- Price$45
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberF-4808
- Product descriptionMLN9708 98%
- Packaging100MG
- Price$90
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product numberX7548
- Product descriptionMLN9708
- Packaging5mg
- Price$170
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product numberX7548
- Product descriptionMLN9708
- Packaging250mg
- Price$420
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberINB0000901
- Product descriptionMLN-9708 95.00%
- Packaging1G
- Price$10065.83
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberINB0000901
- Product descriptionMLN-9708 95.00%
- Packaging10MG
- Price$1006.58
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA4007
- Product descriptionMLN9708
- Packaging50mg
- Price$450
- Updated2026-05-06
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA000QH1 | 4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99% | 1mg | $9 | 2026-05-25 | Buy |
| aablocks | AA000QH1 | 4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99% | 5mg | $20 | 2026-05-25 | Buy |
| aablocks | AA000QH1 | 4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99% | 10mg | $32 | 2026-05-25 | Buy |
| aablocks | AA000QH1 | 4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99% | 25mg | $46 | 2026-05-25 | Buy |
| aablocks | AA000QH1 | 4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 99% | 50mg | $55 | 2026-05-25 | Buy |
| aablocks | AA000QH1 | 4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid 95% | 250mg | $258 | 2026-05-25 | Buy |
| aablocks | AA000QH1 | 4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid ≥98% | 500mg | $435 | 2026-05-25 | Buy |
| aablocks | AA000QH1 | 4-(Carboxymethyl)-2-((R)-1-(2-(2,5-Dichlorobenzamido)Acetamido)-3-Methylbutyl)-6-Oxo-1,3,2-Dioxaborinane-4-Carboxylic Acid ≥98% | 1g | $783 | 2026-05-25 | Buy |
| ACHEMBLOCK | F-4808 | MLN9708 98% | 1G | $495 | 2026-05-27 | Buy |
| ACHEMBLOCK | F-4808 | MLN9708 98% | 25MG | $45 | 2026-05-27 | Buy |
| ACHEMBLOCK | F-4808 | MLN9708 98% | 100MG | $90 | 2026-05-27 | Buy |
| AK Scientific | X7548 | MLN9708 | 5mg | $170 | 2021-12-16 | Buy |
| AK Scientific | X7548 | MLN9708 | 250mg | $420 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | INB0000901 | MLN-9708 95.00% | 1G | $10065.83 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | INB0000901 | MLN-9708 95.00% | 10MG | $1006.58 | 2021-12-16 | Buy |
| ApexBio Technology | A4007 | MLN9708 | 50mg | $450 | 2026-05-06 | Buy |
Properties
Melting point :>227°C (dec.)
Density :1.47
storage temp. :Hygroscopic, -20°C Freezer, Under inert atmosphere
solubility :DMSO (Slightly), Methanol (Slightly, Heated, Sonicated)
pka :1.92±0.20(Predicted)
form :Solid
color :White to Off-White
Density :1.47
storage temp. :Hygroscopic, -20°C Freezer, Under inert atmosphere
solubility :DMSO (Slightly), Methanol (Slightly, Heated, Sonicated)
pka :1.92±0.20(Predicted)
form :Solid
color :White to Off-White
Safety Information
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Description
MLN9708 is an orally bioavailable prodrug of the second-generation proteasome inhibitor MLN2239 . This prodrug rapidly hydrolyzes in plasma to the biologically active form, which inhibits the β5 chymotryptic-like subunit of the 20S proteasome (IC50 = 3.4 nM; Ki = 0.93 nM in cell-free assays). It inhibits the β1 caspase-like and β2 trypsin-like proteolytic sites with IC50 values of 0.03 and 3.5 μM, respectively. MLN9708 has shown antitumor activity both in cell-based assays and in xenograft models and has been examined in phase III clinical trials for potential antimyeloma activity.More related product prices
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