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Elacestrant

Elacestrant Structure
Elacestrant structure
CAS No.
722533-56-4
Chemical Name:
Elacestrant
Synonyms
Elacestrant;Elacestrant (RAD1901);Venadaparib Impurity 54;Elacestrant, 10 mM in DMSO;Elacestrant - API standards;Elacestrant ISO 9001：2015 REACH;inhibit,RAD 1901,Estrogen Receptor/ERR,Inhibitor,Elacestrant,RAD-1901;(R)-6-[2-[Ethyl[4-[2-(ethylamino)ethyl]benzyl]amino]-4-methoxyphenyl]-5,6,7,8-tetrahydronaphthalen-2-ol;(6R)-6-2-ethyl(4-2-(ethylamino)ethylphenylmethyl)amino-4-methoxyphenyl-5,6,7,8-tetrahydronaphthalen-2-ol;2-Naphthalenol, 6-[2-[ethyl[[4-[2-(ethylamino)ethyl]phenyl]methyl]amino]-4-methoxyphenyl]-5,6,7,8-tetrahydro-, (6R)-
CBNumber:
CB63167609
Molecular Formula:
C30H38N2O2
Molecular Weight:
458.63
MDL Number:
MFCD30532693
MOL File:
722533-56-4.mol
MSDS File:
SDS
TDS File:
TDS
Last updated:2026-04-24 16:34:24
Product description Number Pack Size Price
Elacestrant orb611458 5mg $569.5
Elacestrant orb611458 10mg $615.4
Elacestrant orb611458 50mg $1802
Elacestrant >98% DC22559 5mg $280
Elacestrant >98% DC22559 10mg $400
Request For Quotation

Elacestrant Properties

Boiling point 609.5±55.0 °C(Predicted)
Density 1.111±0.06 g/cm3(Predicted)
pka 10.36±0.40(Predicted)
form Solid
color White to off-white
InChIKey SIFNOOUKXBRGGB-AREMUKBSSA-N
SMILES C1=C2C(C[C@H](C3=CC=C(OC)C=C3N(CC)CC3=CC=C(CCNCC)C=C3)CC2)=CC=C1O
FDA UNII FM6A2627A8
NCI Drug Dictionary elacestrant

Elacestrant price

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Biorbyt Ltd orb611458 Elacestrant 722533-56-4 5mg $569.5 2021-12-16 Buy
Biorbyt Ltd orb611458 Elacestrant 722533-56-4 10mg $615.4 2021-12-16 Buy
Biorbyt Ltd orb611458 Elacestrant 722533-56-4 50mg $1802 2021-12-16 Buy
DC Chemicals DC22559 Elacestrant >98% 722533-56-4 5mg $280 2021-12-16 Buy
DC Chemicals DC22559 Elacestrant >98% 722533-56-4 10mg $400 2021-12-16 Buy
Product number Packaging Price Buy
orb611458 5mg $569.5 Buy
orb611458 10mg $615.4 Buy
orb611458 50mg $1802 Buy
DC22559 5mg $280 Buy
DC22559 10mg $400 Buy

Elacestrant Chemical Properties,Uses,Production

Uses

Elacestrant (RAD1901) is an orally available and selective estrogen receptor degrader (SERD) with IC50s of 48 and 870 nM for ERα and ERβ, respectively. Elacestrant also can inhibit growth of ER+ breast cancer cell lines in vitro and in vivo[1][2].

in vivo

Elacestrant (0.3-120 mg/kg; p.o.; single daily for 40 days) antagonizes E2-mediated uterine stimulation in a dose-dependent manner in vivo[1].
Elacestrant (30, 60 mg/kg; p.o.; single daily for 4 weeks) induces complete tumor growth inhibition in mice[2].
Tumor growth inhibition is maintained for 4 weeks after Elacestrant withdrawal[2].

Animal Model:MCF7 cell line xenograft model of mice[2].
Dosage:30, 60 mg/kg
Administration:Oral administration; single daily for 4 weeks.
Result:Inhibited growth of tumor.

References

[1] Garner F, et al. RAD1901: a novel, orally bioavailable selective estrogen receptor degrader that demonstrates antitumor activity in breast cancer xenograft models. Anticancer Drugs. 2015 Oct;26(9):948-56. DOI:10.1097/CAD.0000000000000271
[2] Bihani T, et al. Elacestrant (RAD1901), a Selective Estrogen Receptor Degrader (SERD), Has Antitumor Activity in Multiple ER+ Breast Cancer Patient-derived Xenograft Models. Clin Cancer Res. 2017 Aug 15;23(16):4793-4804. DOI:10.1158/1078-0432.CCR-16-2561

Elacestrant Preparation Products And Raw materials

Raw materials

Preparation Products

Elacestrant Suppliers

Global( 90)Suppliers
Supplier Tel Email Country ProdList Advantage
ATK CHEMICAL COMPANY LIMITED 		+undefined-21-51877795 ivan@atkchemical.com China 33024 60
Jinan Carbotang Biotech Co.,Ltd. 		+8615866703830 figo.gao@foxmail.com China 8497 58
BOC Sciences 		+1-631-485-4226 inquiry@bocsci.com United States 19552 58
CONIER CHEM AND PHARMA LIMITED 		+8618523575427 sales@conier.com China 49977 58
TargetMol Chemicals Inc. 		+1-781-999-5354; +17819995354 marketing@targetmol.com United States 32467 58
Dideu Industries Group Limited 		+86-29-89586680 +86-15129568250 1026@dideu.com China 18895 58
Zhejiang J&C Biological Technology Co.,Limited 		+1-2135480471 +1-2135480471; sales@sarms4muscle.com China 10473 58
TargetMol Chemicals Inc. 		+1-781-999-5354; support@targetmol.com United States 39040 58
Chemtour Biotech Co., Ltd 		+8617327281506 market@chemtour.com China 1521 58
Wuhan Topule Biopharmaceutical Co., Ltd 		+8618327326525 masar@topule.com China 8467 58
Supplier Advantage
ATK CHEMICAL COMPANY LIMITED 		60
Jinan Carbotang Biotech Co.,Ltd. 		58
BOC Sciences 		58
CONIER CHEM AND PHARMA LIMITED 		58
TargetMol Chemicals Inc. 		58
Dideu Industries Group Limited 		58
Zhejiang J&C Biological Technology Co.,Limited 		58
TargetMol Chemicals Inc. 		58
Chemtour Biotech Co., Ltd 		58
Wuhan Topule Biopharmaceutical Co., Ltd 		58

View Lastest Price from Elacestrant manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
Elacestrant pictures 2026-04-24 Elacestrant
722533-56-4
 US $126.00-396.00 / mg 99.92% 10g TargetMol Chemicals Inc.
Elacestrant pictures 2026-04-24 Elacestrant
722533-56-4
 US $126.00-396.00 / mg 99.92% 10g TargetMol Chemicals Inc.
  • Elacestrant pictures
  • Elacestrant
    722533-56-4
  • US $126.00-396.00 / mg
  • 99.92%
  • TargetMol Chemicals Inc.
  • Elacestrant pictures
  • Elacestrant
    722533-56-4
  • US $126.00-396.00 / mg
  • 99.92%
  • TargetMol Chemicals Inc.

Elacestrant Spectrum

Elacestrant(722533-56-4)1HNMR

722533-56-4(Elacestrant)Related Search:

Fulvestrant ESTETROL β-Estradiol Elacestrant dihydrochloride 2-Naphthalenol, 6-(2-amino-4-methoxyphenyl)-5,6,7,8-tetrahydro-, (6R)-
Acetamide, N-[2-[3,4-dihydro-6-(phenylmethoxy)-2-naphthalenyl]-5-methoxyphenyl]- Acetamide, N-[5-methoxy-2-(1,2,3,4-tetrahydro-6-hydroxy-2-naphthalenyl)phenyl]-

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Elacestrant Elacestrant (RAD1901) 2-Naphthalenol, 6-[2-[ethyl[[4-[2-(ethylamino)ethyl]phenyl]methyl]amino]-4-methoxyphenyl]-5,6,7,8-tetrahydro-, (6R)- Elacestrant ISO 9001：2015 REACH inhibit,RAD 1901,Estrogen Receptor/ERR,Inhibitor,Elacestrant,RAD-1901 (6R)-6-2-ethyl(4-2-(ethylamino)ethylphenylmethyl)amino-4-methoxyphenyl-5,6,7,8-tetrahydronaphthalen-2-ol (R)-6-[2-[Ethyl[4-[2-(ethylamino)ethyl]benzyl]amino]-4-methoxyphenyl]-5,6,7,8-tetrahydronaphthalen-2-ol Venadaparib Impurity 54 Elacestrant - API standards Elacestrant, 10 mM in DMSO (6R)-6-{2-[Ethyl({4-[2-(ethylamino)ethyl]phenyl}methyl)amino]-4-methoxyphenyl}-5,6,7,8-tetrahydronaphthalen-2-ol. dihydrochloride 722533-56-4 22533-56-4 API