ガベキサート 化学特性,用途語,生産方法
効能
抗凝固薬, 血漿カリクレイン阻害薬
使用
Gabexate mesylate is used in combination with somatostatin and octreotide in the treatment of severe acute pancreatitis in elderly patients.
生物活性
Serine protease inhibitor; inhibits trypsin, plasmin, plasma kallikrein and thrombin (IC 50 values are 9.4, 30, 41 and 110 mM respectively). Antithrombotic in vitro and in vivo . Also inhibits LPS-induced TNF- α production, probably by inhibiting NF- κ B and AP-1 activation.
ガベキサート 上流と下流の製品情報
原材料
準備製品