ChemicalBook >> CAS DataBase List >>Paliperidone Palmitate
Paliperidone Palmitate
- CAS No.
- 199739-10-1
- Chemical Name:
- Paliperidone Palmitate
- Synonyms
- Invega Sustenna;RO 92670;Paliperidone Palmitate;Paliperidone Palmitate-d31;Paliperidone Palmitate [USAN];9-Hydroxyrisperidone palmitate;Paliperidone Palmitate USP/EP/BP;Paliperidone Palmitate Benzisoxazole Impurity;Paliperidone Impurity 39 (Paliperidone Palmitate);3-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-9-yl palmitate
- CBNumber:
- CB82519012
- Molecular Formula:
- C39H57FN4O4
- Molecular Weight:
- 664.89
- MDL Number:
- MFCD24386477
- MOL File:
- 199739-10-1.mol
- MSDS File:
- SDS
Last updated:2024-04-22 13:56:47
| Melting point | 110-115°C |
|---|---|
| Boiling point | 736.3±70.0 °C(Predicted) |
| Density | 1.19 |
| storage temp. | Sealed in dry,Store in freezer, under -20°C |
| solubility | Chloroform (Slightly), Ethyl Acetate (Slightly, Heated, Sonicated), Methanol (Slightly) |
| form | Solid |
| pka | 8.07±0.10(Predicted) |
| color | Off-White to Light Beige |
| FDA UNII | R8P8USM8FR |
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS06 |
|---|---|
| Signal word | Danger |
| Hazard statements | H301 |
| Precautionary statements | P264-P270-P301+P310-P321-P330-P405-P501 |
Paliperidone Palmitate price More Price(11)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| TRC | P141020 | PaliperidonePalmitate | 199739-10-1 | 500mg | $210 | 2021-12-16 | Buy |
| Activate Scientific | AS148096 | PaliperidonePalmitate 98% | 199739-10-1 | 250mg | $233 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0027470 | PALIPERIDONE PALMITATE 95.00% | 199739-10-1 | 25MG | $750.75 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0027470 | PALIPERIDONE PALMITATE 95.00% | 199739-10-1 | 250MG | $1963.5 | 2021-12-16 | Buy |
| ChemScene | CS-0016387 | Paliperidonepalmitate 98.16% | 199739-10-1 | 10mg | $70 | 2021-12-16 | Buy |
Paliperidone Palmitate Chemical Properties,Uses,Production
Description
Paliperidone palmitate is an atypical long acting antipsychotics，which can fast onset in acute phase and continuously improve the symptoms in maintenance phase． It has the solid efficacy and convenient ad[1]ministration，which offer a new option for schizophrenia treatment and will help patients to adhere the treatment and prevent relapse． As the sole long acting antipsychotics with monthly injection，it was approved by CFDA in 2011 and indicated for the acute and maintenance treatment of schizophrenia．
Uses
Paliperidone Palmitate is a long-acting injectable atypical antipsychotic used in the treatment of schizophrenia.
Definition
ChEBI: 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2-methyl-4-oxo-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-9-yl hexadecanoate is a fatty acid ester obtained by the formal condensation of the carboxy group of hexadecanoic acid with the hydroxy group of 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-9-hydroxy-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one. It is a member of 1,2-benzoxazoles, a heteroarylpiperidine, an organofluorine compound, a pyridopyrimidine and a fatty acid ester.
Side effects
The review of the literature also underlined that paliperidone palmitate is well tolerated, compared with placebo. Frequency and severity of side-effects such as extrapyramidal symptoms, hyperprolactinemia and weight gain, was similar or less than those found in treatment with other atypical antipsychotics, including long-acting ones.
Paliperidone Palmitate Preparation Products And Raw materials
Raw materials
Preparation Products
Global( 211)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Jewim Pharmaceutical (Shandong) Co., Ltd. | +86-15552509998 +86-15621883869 | liutf@jewim.com.cn | China | 251 | 58 |
| Hebei Mojin Biotechnology Co., Ltd | +8613288715578 | sales@hbmojin.com | China | 12456 | 58 |
| Sinoway Industrial co., ltd. | 0592-5800732; +8613806035118 | xie@china-sinoway.com | China | 992 | 58 |
| Henan Bao Enluo International TradeCo.，LTD | +86-17331933971 +86-17331933971 | deasea125996@gmail.com | China | 2503 | 58 |
| Zibo Hangyu Biotechnology Development Co., Ltd | +86-0533-2185556 +8617865335152 | Mandy@hangyubiotech.com | China | 11013 | 58 |
| Ouhuang Engineering Materials (Hubei) Co., Ltd | +8617702722807 | admin@hbouhuang.com | China | 2259 | 58 |
| Capot Chemical Co.,Ltd. | 571-85586718 +8613336195806 | sales@capotchem.com | China | 29797 | 60 |
| Hangzhou FandaChem Co.,Ltd. | 008657128800458; +8615858145714 | fandachem@gmail.com | China | 9348 | 55 |
| Lianyungang happen teng technology co., LTD | 15950718863 | wang666xt@163.com | CHINA | 295 | 58 |
| career henan chemical co | +86-0371-86658258 | sales@coreychem.com | China | 29914 | 58 |
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View Lastest Price from Paliperidone Palmitate manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2024-04-22 | Paliperidone Palmitate
199739-10-1
|
US $50.00 / kg | 1kg | 99.10% | 50000kg | Ouhuang Engineering Materials (Hubei) Co., Ltd | |
 |
2024-04-22 | Paliperidone Palmitate
199739-10-1
|
US $175.00-85.00 / Kg/Bag | 1Kg/Bag | 0.99 | 20 tons | Sinoway Industrial co., ltd. | |
 |
2024-01-02 | Paliperidone Palmitate
199739-10-1
|
US $70.00-700.00 / kg | 10kg | 0.99 | 20tons | Zibo Hangyu Biotechnology Development Co., Ltd |
-
- Paliperidone Palmitate
199739-10-1
- US $50.00 / kg
- 99.10%
- Ouhuang Engineering Materials (Hubei) Co., Ltd
-
- Paliperidone Palmitate
199739-10-1
- US $175.00-85.00 / Kg/Bag
- 0.99
- Sinoway Industrial co., ltd.
-
- Paliperidone Palmitate
199739-10-1
- US $70.00-700.00 / kg
- 0.99
- Zibo Hangyu Biotechnology Development Co., Ltd
199739-10-1(Paliperidone Palmitate)Related Search:
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din-9-yl hexadecanoate
Hexadecanoic acid 3-[2-[4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl]-ethyl]-6,7,8,9-tetrahydro-2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl ester
Paliperidone Palmitate
Paliperidone Palmitate [USAN]
RO 92670
9-Hydroxyrisperidone palmitate
Hexadecanoic acid 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl ester
Paliperidone Palmitate-d31
Paliperidone Impurity 39 (Paliperidone Palmitate)
3-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethyl)-2-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-9-yl palmitate
Paliperidone Palmitate USP/EP/BP
Paliperidone palmitateQ: What is
Paliperidone palmitate Q: What is the CAS Number of
Paliperidone palmitate Q: What is the storage condition of
Paliperidone palmitate Q: What are the applications of
Paliperidone palmitate
Invega Sustenna
Paliperidone Palmitate Benzisoxazole Impurity
199739-10-1
C39H57FN4O4
Heterocycles
Intermediates & Fine Chemicals
Pharmaceuticals
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