ChemicalBook >> CAS DataBase List >>SB 242084 (hydrochloride)

SB 242084 (hydrochloride)

CAS No.
1049747-87-6
Chemical Name:
SB 242084 (hydrochloride)
Synonyms
SB 242084 2HCL;CAS 1049747-87-6;SB-242084 HCl salt;SB 242084 (hydrochloride);SB242084;SB 242084;CAS 1049747-87-6
CBNumber:
CB82592406
Molecular Formula:
C21H21Cl3N4O2
Molecular Weight:
467.77604
MDL Number:
MOL File:
1049747-87-6.mol
MSDS File:
SDS
Last updated:2023-06-30 15:45:59

SB 242084 (hydrochloride) Properties

storage temp. Sealed in dry,Room Temperature
solubility Ethanol:1.0(Max Conc. mg/mL);2.14(Max Conc. mM)
PBS (pH 7.2):10.0(Max Conc. mg/mL);21.38(Max Conc. mM)
DMSO:59.63(Max Conc. mg/mL);127.47(Max Conc. mM)
DMF:30.0(Max Conc. mg/mL);64.13(Max Conc. mM)
form A crystalline solid

SAFETY

Risk and Safety Statements

Symbol(GHS)  GHS hazard pictograms
GHS07
Signal word  Warning
Hazard statements  H315-H319-H335
Precautionary statements  P261-P264-P271-P280-P302+P352-P304+P340-P305+P351+P338-P312-P321-P362+P364-P332+P313-P337+P313-P403+P233-P405-P501
NFPA 704
0
2 0

SB 242084 (hydrochloride) price More Price(14)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Cayman Chemical 10096 SB-242084 (hydrochloride) ≥98% 1049747-87-6 1mg $47 2024-03-01 Buy
Cayman Chemical 10096 SB-242084 (hydrochloride) ≥98% 1049747-87-6 5mg $137 2024-03-01 Buy
Cayman Chemical 10096 SB-242084 (hydrochloride) ≥98% 1049747-87-6 10mg $182 2024-03-01 Buy
TRC S155020 SB242084Hydrochloride 1049747-87-6 1mg $85 2021-12-16 Buy
Usbiological 465901 SB 242084 Hydrochloride 1049747-87-6 1mg $360 2021-12-16 Buy
Product number Packaging Price Buy
10096 1mg $47 Buy
10096 5mg $137 Buy
10096 10mg $182 Buy
S155020 1mg $85 Buy
465901 1mg $360 Buy

SB 242084 (hydrochloride) Chemical Properties,Uses,Production

Description

Serotonin (5-hydroxytryptamine, 5-HT) is a neurotransmitter that activates specific receptors located primarily in the gut and central nervous system. SB-242084 is an antagonist of the 5-HT2C receptor (pKi = 9.0), with at least 100-fold more selectivity over other 5-HT, dopamine, or adrenergic receptors. In vivo, it is brain penetrant and has significant anxiolytic activity, without sedative, proconvulsant, or hyperphagic properties. SB-242084 has been used extensively in animal research to evaluate, for example, 5-HT2C receptor agonists and neurotransmitter receptor interactions in mice.

Uses

SB 242084 Hydrochloride is an antagonist of the SR-2C.

Definition

ChEBI: 6-chloro-5-methyl-N-[6-(2-methylpyridin-3-yl)oxypyridin-3-yl]-2,3-dihydroindole-1-carboxamide;dihydrochloride is an organic molecular entity, an indole alkaloid and a pyridine. It has a role as a receptor modulator.

storage

Desiccate at +4°C

SB 242084 (hydrochloride) Preparation Products And Raw materials

Raw materials

Preparation Products

SB 242084 (hydrochloride) Suppliers

Global( 60)Suppliers
Supplier Tel Email Country ProdList Advantage
HANGZHOU CLAP TECHNOLOGY CO.,LTD
86-571-88216897,88216896 13588875226 sales@hzclap.com CHINA 6313 58
InvivoChem
+1-708-310-1919 +1-13798911105 sales@invivochem.cn United States 6393 58
Nantong HI-FUTURE Biology Co., Ltd.
+undefined18051384581 sales@chemhifuture.com China 3136 58
Wuhan Topule Biopharmaceutical Co., Ltd
+8618327326525 masar@topule.com China 8474 58
Aladdin Scientific
+1-833-552-7181 sales@aladdinsci.com United States 57511 58
Amadis Chemical Company Limited
571-89925085 sales@amadischem.com China 131981 58
Shanghai Aladdin Bio-Chem Technology Co.,LTD 400-6206333 18521732826; market@aladdin-e.com China 25015 65
MedChemexpress LLC 021-58955995 sales@medchemexpress.cn United States 4863 58
ShangHai Biochempartner Co.,Ltd 17754423994 17754423994 2853530910@QQ.com China 8011 62
Musechem +1-800-259-7612 info@musechem.com United States 4662 60
SB 242084 (hydrochloride) SB-242084 HCl salt CAS 1049747-87-6 SB242084;SB 242084;CAS 1049747-87-6 SB 242084 2HCL 1049747-87-6 C21H19ClN4O22ClHH2O API