Chlormezanone improves the emotional state of the patient, relieving moderate anxiety
and stress. However, it has a number of side effects, and because it does not have any
advantage over other anxiolytics, it is rarely used in practice.
정의
ChEBI: A 1,3-thiazine that is 1,3-thiazinan-4-one S,S-dioxide in which a hydrogen at position 2 is substituted by a 4-chlorophenyl group and the hydrogen attached to the nitrogen is substituted by methyl. A non-benzodiazepine
muscle relaxant, it was used in the management of anxiety and in the treatment of muscle spasms until being discontinued worldwide by its manufacturer in 1996, due to rare but serious cutaneous reactions.
World Health Organization (WHO)
Chlormezanone is a sedative with antianxiety properties and a
central skeletal muscle relaxant effect. It had already been falling into
obsolescence for several years.
생물학적 활성
Anxiolytic and skeletal muscle relaxant that acts at the benzodiazepine site of GABA A receptors.