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Ketanserin

CAS No.
74050-98-9
Chemical Name:
Ketanserin
Synonyms
RHS;Ket;p73L;p73H;OFC8;EEC3;SHFM4;p53CP;TP53L;TP73L
CBNumber:
CB5704758
Molecular Formula:
C22H22FN3O3
Molecular Weight:
395.43
MDL Number:
MFCD00083392
MOL File:
74050-98-9.mol
Last updated:2024-10-31 18:15:48

Ketanserin Properties

Melting point 227-235°C
Density 1.280±0.06 g/cm3(Predicted)
storage temp. Sealed in dry,2-8°C
solubility DMF: 10 mg/mL, clear, colorless
form Solid
pka 7.5(at 25℃)
color White to Off-White
Merck 14,5296
CAS DataBase Reference 74050-98-9(CAS DataBase Reference)
FDA UNII 97F9DE4CT4
ATC code C02KD01

SAFETY

Risk and Safety Statements

Symbol(GHS)  GHS hazard pictograms
GHS07
Signal word  Warning
Hazard statements  H302
Precautionary statements  P501-P270-P264-P301+P312+P330
WGK Germany  3
RTECS  VA1411190
HS Code  29339900
NFPA 704
0
2 0

Ketanserin price More Price(25)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
TCI Chemical K0051 Ketanserin >98.0%(HPLC)(T) 74050-98-9 200mg $62 2024-03-01 Buy
TCI Chemical K0051 Ketanserin >98.0%(HPLC)(T) 74050-98-9 1g $186 2024-03-01 Buy
TRC K165450 Ketanserin 74050-98-9 250mg $135 2021-12-16 Buy
TRC K165450 Ketanserin 74050-98-9 50mg $50 2021-12-16 Buy
ChemScene CS-6055 Ketanserin 98.57% 74050-98-9 50mg $50 2021-12-16 Buy
Product number Packaging Price Buy
K0051 200mg $62 Buy
K0051 1g $186 Buy
K165450 250mg $135 Buy
K165450 50mg $50 Buy
CS-6055 50mg $50 Buy

Ketanserin Chemical Properties,Uses,Production

Description

Ketanserin is an antihypertensive agent with antagonist properties at both the serotonin-S2 and α1-adrenergic receptors. Its mechanism of action, while still controversial, may involve interactions at both of these loci.

Chemical Properties

Off-White Solid

Originator

Janssen (Belgium)

Uses

An antihypertensive, with affinity for multiple GPCR receptors.

Uses

receptor antagonist

Definition

ChEBI: A member of the class of quinazolines that is quinazoline-2,4(1H,3H)-dione which is substituted at position 3 by a 2-[4-(p-fluorobenzoyl)piperidin-1-yl]ethyl group.

brand name

SEREFREX

Purification Methods

It has been purified by recrystallisation from 4-methyl-3-pentanone [Peeters et al. Cryst Structure Commun 11 375 1982, Kacprowicz et al. J Chromatogr 272 417 1983, Davies et al. J Chromatogr 275 232 1983]. It is an antihypertensive.

Ketanserin Preparation Products And Raw materials

Raw materials

Preparation Products

Global( 226)Suppliers
Supplier Tel Email Country ProdList Advantage
Hebei Yanxi Chemical Co., Ltd.
+8617531190177 peter@yan-xi.com China 5858 58
Hebei Weibang Biotechnology Co., Ltd
+8617732866630 bess@weibangbio.com China 18232 58
Henan Tianfu Chemical Co.,Ltd.
+86-0371-55170693 +86-19937530512 info@tianfuchem.com China 21639 55
ATK CHEMICAL COMPANY LIMITED
+undefined-21-51877795 ivan@atkchemical.com China 32820 60
career henan chemical co
+86-0371-86658258 +8613203830695 sales@coreychem.com China 29886 58
Hubei xin bonus chemical co. LTD
86-13657291602 linda@hubeijusheng.com CHINA 22963 58
Shandong chuangyingchemical Co., Ltd.
18853181302 sale@chuangyingchem.com CHINA 5906 58
Chongqing Chemdad Co., Ltd
+86-023-6139-8061 +86-86-13650506873 sales@chemdad.com China 39894 58
CONIER CHEM AND PHARMA LIMITED
+8618523575427 sales@conier.com China 49374 58
Zhengzhou Alfa Chemical Co.,Ltd
+8618530059196 sale04@alfachem.cn China 13486 58

View Lastest Price from Ketanserin manufacturers

Image Update time Product Price Min. Order Purity Supply Ability Manufacturer
Ketanserin pictures 2024-10-31 Ketanserin
74050-98-9
US $30.00-88.00 / mg 99.73% 10g TargetMol Chemicals Inc.
Ketanserin pictures 2024-10-31 Ketanserin
74050-98-9
US $30.00-88.00 / mg 99.73% 10g TargetMol Chemicals Inc.
Ketanserin pictures 2024-10-31 Ketanserin
74050-98-9
US $0.00 / Kg/Bag 2Kg/Bag 99% up / EP 20 tons Sinoway Industrial co., ltd.
  • Ketanserin pictures
  • Ketanserin
    74050-98-9
  • US $30.00-88.00 / mg
  • 99.73%
  • TargetMol Chemicals Inc.
  • Ketanserin pictures
  • Ketanserin
    74050-98-9
  • US $30.00-88.00 / mg
  • 99.73%
  • TargetMol Chemicals Inc.
  • Ketanserin pictures
  • Ketanserin
    74050-98-9
  • US $0.00 / Kg/Bag
  • 99% up / EP
  • Sinoway Industrial co., ltd.

Ketanserin Spectrum

B(p51A) B(p51B) EEC3 OFC8 p53CP p63, GST tagged human p73H p73L RHS SHFM4 TP53CP TP53L TP73L 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-2,4[1h,3h]-quinazolinedione KETANSERIN 3-(2-(4-(4-fluorobenzoyl)piperidin-1-yl)ethyl)quinazoline-2,4(1H,3H)-dione 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4-(IH,3H)-quinazolinedione Ketanserin (Vulketan Gel)| Ketanserin(R 41 468) Ket Ketensin Perketan R-49945 Serefrex Serepress Sufrexal Taseron 2,4(1H,3H)-Quinazolinedione, 3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]- 3-[2-[4-(4-Fluorobenzoyl)piperidin-1-yl]ethyl]-1H-quinazoline-2,4-dione 3-[2-[4-(4-Fluorobenzoyl)piperidin-1-yl]ethyl]-2,4(1H,3H)-quinazolinedione 3-[2-[4-(4-Fluorobenzoyl)piperidino]ethyl]-2,4(1H,3H)-quinazolinedione Ketanserine Ketanserin, 99%, a specific 5-HT2A serotonin receptor antagonist Ketanserin> Ketanserinum Ketanserin USP/EP/BP Ketanserine Base 3-{2-[4-(4-fluorobenzoyl)piperidin-1-yl]ethyl}-1,2,3, 4-tetrahydroquinazoline-2,4-dione TIANFU CHEM----Ketanserin Ketanserin,3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4[1H,3H]-quinazolinedione 3-[2-[4-(4-Fluorobenzoyl)-1-piperidyl]ethyl]quinazoline-2,4(1H,3H)-dione 74050-98-9 C22H22FN3O3 Intermediates & Fine Chemicals Pharmaceuticals Other APIs ketone