イミダプリル 化学特性,用途語,生産方法
用途
ACE阻害薬降圧効果
効能
血圧降下薬, アンジオテンシン変換酵素(ACE)阻害薬
説明
Imidapril is a new ACE inhibitor launched in Japan as a once-daily therapy for
hypertension. Its active metabolite has more potent inhibitory effects on all tissue ACES from
spontaneously hypertensive rats (SHRs) and Wistar Kyoto rats (WKYs) than many other ACE
inhibitors including enalapril and captopril. It has a very long duration of action. In strokeprone
spontaneously hypertensive rats (SHRSP), imidapril is effective in stroke prevention at
a considerably lower dose than enalapril. This stroke preventive effect has been suggested to
be primarily by an indirect mechanism related to the amelioration of kidney dysfunction.
化学的特性
White Solid
使用
Angiotensin converting enzyme (ACE) inhibitor. Antihypertensive
イミダプリル 上流と下流の製品情報
原材料
準備製品