ERK Inhibitor
- CAS No.
- 1049738-54-6
- Chemical Name:
- ERK Inhibitor
- Synonyms
- ERK-IN-4;ERK Inhibitor - CAS 1049738-54-6 - Calbiochem;3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylene]-2,4-thiazolidinedione,monohydrochloride;(5Z)-3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione:hydrochloride
- CBNumber:
- CB13136749
- Molecular Formula:
- C14H17ClN2O3S
- Molecular Weight:
- 328.81
- MDL Number:
- MFCD09038681
- MOL File:
- 1049738-54-6.mol
ERK Inhibitor price More Price(4)
Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|---|
Cayman Chemical | 15944 | ERK Inhibitor ≥95% | 1049738-54-6 | 500μg | $32 | 2024-03-01 | Buy |
Cayman Chemical | 15944 | ERK Inhibitor ≥95% | 1049738-54-6 | 1mg | $50 | 2024-03-01 | Buy |
Cayman Chemical | 15944 | ERK Inhibitor ≥95% | 1049738-54-6 | 5mg | $117 | 2024-03-01 | Buy |
AK Scientific | 9473CW | ErkInhibitor | 1049738-54-6 | 5mg | $228 | 2021-12-16 | Buy |
ERK Inhibitor Chemical Properties,Uses,Production
Description
ERK inhibitor is a cell-
General Description
A cell-permeable and reversible thiazolidinedione compound that displays anti-proliferative properties (IC50 ≤ 25 μM in HeLa, A549, and SUM-159 tumor cells). Preferentially binds to ERK2 with a KD of ~5 μM and prevents its interaction with protein substrates. Shown to block ERK-mediated phosphorylation of ribosomal S6 kinase-1 (RSK-1) and ternary complex factor Elk-1 in HeLa cells, while exhibiting little effect on ERK1/2 phosphorylation by MEK1/2.
Biochem/physiol Actions
Primary TargetERK
ERK Inhibitor Preparation Products And Raw materials
Raw materials
Preparation Products
ERK Inhibitor Suppliers
Supplier | Tel | Country | ProdList | Advantage | |
---|---|---|---|---|---|
Shaanxi Cuikang Pharmaceutical Technology Co., Ltd | +8618829768577 | gao490372054@gamil.com | China | 1250 | 58 |
Wuhan Topule Biopharmaceutical Co., Ltd | +8618327326525 | masar@topule.com | China | 8474 | 58 |
Shaanxi Cuikang Pharmaceutical Technology Co., Ltd | +86-18791163155 +86-13119157289 | 13119157289@163.com | China | 2972 | 58 |
Aladdin Scientific | +1-+1(833)-552-7181 | sales@aladdinsci.com | United States | 57511 | 58 |
Shanghai Run-Biotech Co., Ltd. | 021-57171705 13817537615 | sales@run-biotech.com | China | 2484 | 58 |
Sigma-Aldrich | 021-61415566 800-8193336 | orderCN@merckgroup.com | China | 51471 | 80 |
BOC Sciences | 16314854226 | info@bocsci.com | United States | 9926 | 65 |
Shanghai EFE Biological Technology Co., Ltd. | 021-65675885 18964387627 | info@efebio.com | China | 9707 | 58 |
Shanghai Hongye Biotechnology Co. Ltd | 400-9205774 | sales@glpbio.cn | China | 6870 | 58 |
ChemeGen(Shanghai) Biotechnology Co.,Ltd. | 18818260767 | sales@chemegen.com | China | 11289 | 58 |